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- [1] Discovery of an Oral Respiratory Syncytial Virus (RSV) Fusion Inhibitor (GS-5806) and Clinical Proof of Concept in a Human RSV Challenge StudyJOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (04) : 1630 - 1643Mackman, Richard L.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USASangi, Michael论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USASperandio, David论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USAParrish, Jay P.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USAEisenberg, Eugene论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USAPerron, Michel论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USAHui, Hon论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USAZhang, Lijun论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USASiegel, Dustin论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USAYang, Hai论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USASaunders, Oliver论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USABoojamra, Constantine论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USALee, Gary论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USASamuel, Dharmaraj论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USABabaoglu, Kerim论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USACarey, Anne论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USAGilbert, Brian E.论文数: 0 引用数: 0 h-index: 0机构: Baylor Coll Med, Dept Mol Virol & Microbiol, Houston, TX 77030 USA Gilead Sci, Foster City, CA 94404 USAPiedra, Pedro A.论文数: 0 引用数: 0 h-index: 0机构: Baylor Coll Med, Dept Mol Virol & Microbiol, Houston, TX 77030 USA Gilead Sci, Foster City, CA 94404 USAStrickley, Robert论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USAIwata, Quynh论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USAHayes, Jaclyn论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USAStray, Kirsten论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USAKinkade, April论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USATheodore, Dorothy论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USAJordan, Robert论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USADesai, Manoj论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USACihlar, Tomas论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA 94404 USA Gilead Sci, Foster City, CA 94404 USA
- [2] Oral GS-5806 Activity in a Respiratory Syncytial Virus Challenge StudyNEW ENGLAND JOURNAL OF MEDICINE, 2014, 371 (08): : 711 - 722DeVincenzo, John P.论文数: 0 引用数: 0 h-index: 0机构: Univ Tennessee, Sch Med, Memphis, TN USA Childrens Fdn Res Inst, Le Bonheur Childrens Hosp, Memphis, TN 38103 USA Univ Tennessee, Sch Med, Memphis, TN USAWhitley, Richard J.论文数: 0 引用数: 0 h-index: 0机构: Univ Alabama Birmingham, Sch Med, Birmingham, AL USA Univ Tennessee, Sch Med, Memphis, TN USAMackman, Richard L.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Univ Tennessee, Sch Med, Memphis, TN USAScaglioni-Weinlich, Cecilia论文数: 0 引用数: 0 h-index: 0机构: Univ Tennessee, Sch Med, Memphis, TN USA Univ Tennessee, Sch Med, Memphis, TN USAHarrison, Lisa论文数: 0 引用数: 0 h-index: 0机构: Univ Tennessee, Sch Med, Memphis, TN USA Univ Tennessee, Sch Med, Memphis, TN USAFarrell, Eric论文数: 0 引用数: 0 h-index: 0机构: Univ Tennessee, Sch Med, Memphis, TN USA Univ Tennessee, Sch Med, Memphis, TN USAMcBride, Stephen论文数: 0 引用数: 0 h-index: 0机构: Univ Tennessee, Sch Med, Memphis, TN USA Univ Tennessee, Sch Med, Memphis, TN USALambkin-Williams, Robert论文数: 0 引用数: 0 h-index: 0机构: Retroscreen Virol, London, England Univ Tennessee, Sch Med, Memphis, TN USAJordan, Robert论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Univ Tennessee, Sch Med, Memphis, TN USAXin, Yan论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Univ Tennessee, Sch Med, Memphis, TN USARamanathan, Srini论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Univ Tennessee, Sch Med, Memphis, TN USAO'Riordan, Thomas论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Univ Tennessee, Sch Med, Memphis, TN USALewis, Sandra A.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Univ Tennessee, Sch Med, Memphis, TN USALi, Xiaoming论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Univ Tennessee, Sch Med, Memphis, TN USAToback, Seth L.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Univ Tennessee, Sch Med, Memphis, TN USALin, Shao-Lee论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Univ Tennessee, Sch Med, Memphis, TN USAChien, Jason W.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Univ Tennessee, Sch Med, Memphis, TN USA
- [3] A mechanistic model describing the effect of respiratory syncytial virus (RSV) kinetics on clinical symptom score, and disease attenuation by presatovir (GS-5806)JOURNAL OF PHARMACOKINETICS AND PHARMACODYNAMICS, 2016, 43 : S64 - S64Lutz, Justin D.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Dept Clin Pharmacol, 353 Lakeside Dr, Foster City, CA 94404 USA Gilead Sci Inc, Dept Clin Pharmacol, 353 Lakeside Dr, Foster City, CA 94404 USAPatel, Kashyap论文数: 0 引用数: 0 h-index: 0机构: D3 Med, Parsippany, NJ USA Gilead Sci Inc, Dept Clin Pharmacol, 353 Lakeside Dr, Foster City, CA 94404 USASmith, Patrick论文数: 0 引用数: 0 h-index: 0机构: D3 Med, Parsippany, NJ USA Gilead Sci Inc, Dept Clin Pharmacol, 353 Lakeside Dr, Foster City, CA 94404 USAChien, Jason W.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Dept Clin Res, 353 Lakeside Dr, Foster City, CA 94404 USA Gilead Sci Inc, Dept Clin Pharmacol, 353 Lakeside Dr, Foster City, CA 94404 USAJordan, Robert论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Dept Biol, 353 Lakeside Dr, Foster City, CA 94404 USA Gilead Sci Inc, Dept Clin Pharmacol, 353 Lakeside Dr, Foster City, CA 94404 USAXin, Yan论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Dept Clin Pharmacol, 353 Lakeside Dr, Foster City, CA 94404 USA Gilead Sci Inc, Dept Clin Pharmacol, 353 Lakeside Dr, Foster City, CA 94404 USARamanathan, Srini论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Dept Clin Pharmacol, 353 Lakeside Dr, Foster City, CA 94404 USA Gilead Sci Inc, Dept Clin Pharmacol, 353 Lakeside Dr, Foster City, CA 94404 USAMathias, Anita论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Dept Clin Pharmacol, 353 Lakeside Dr, Foster City, CA 94404 USA Gilead Sci Inc, Dept Clin Pharmacol, 353 Lakeside Dr, Foster City, CA 94404 USA
- [4] A Phase 2b, Randomized, Double-Blind, Placebo-Controlled Trial of Presatovir (GS-5806), a Novel Oral RSV Fusion Inhibitor, for the Treatment of Respiratory Syncytial Virus (RSV) in Hospitalized AdultsAMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE, 2018, 197Hanfelt-Goade, D.论文数: 0 引用数: 0 h-index: 0机构: Tauranga Hosp, Internal Med, Tauranga, New Zealand Tauranga Hosp, Internal Med, Tauranga, New ZealandMaimon, N.论文数: 0 引用数: 0 h-index: 0机构: Soroka Univ, Med Ctr, Beer Sheva, Israel Tauranga Hosp, Internal Med, Tauranga, New ZealandNimer, A.论文数: 0 引用数: 0 h-index: 0机构: Galilee Med Ctr, Nahariyya, Israel Tauranga Hosp, Internal Med, Tauranga, New ZealandRiviere, F.论文数: 0 引用数: 0 h-index: 0机构: Hop Instruct Armees Percy, Clamart, France Tauranga Hosp, Internal Med, Tauranga, New ZealandCatherinot, E.论文数: 0 引用数: 0 h-index: 0机构: Hop Foch, Suresnes, France Tauranga Hosp, Internal Med, Tauranga, New ZealandIson, M.论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Chicago, IL 60611 USA Tauranga Hosp, Internal Med, Tauranga, New ZealandJeong, S.论文数: 0 引用数: 0 h-index: 0机构: Gachon Univ Gil Med Ctr, Incheon, South Korea Tauranga Hosp, Internal Med, Tauranga, New Zealand论文数: 引用数: h-index:机构:Gafter-Gvili, A.论文数: 0 引用数: 0 h-index: 0机构: Rabin Med Ctr, Petah Tiqwa, Israel Tauranga Hosp, Internal Med, Tauranga, New ZealandNama, S.论文数: 0 引用数: 0 h-index: 0机构: Gold Coast Univ Hosp, Southport, Qld, Australia Tauranga Hosp, Internal Med, Tauranga, New ZealandNapora, P.论文数: 0 引用数: 0 h-index: 0机构: Ctr Badan Klin, Wroclaw, Poland Tauranga Hosp, Internal Med, Tauranga, New ZealandChowers, M.论文数: 0 引用数: 0 h-index: 0机构: Meir Med Ctr, Kefar Sava, Israel Tauranga Hosp, Internal Med, Tauranga, New ZealandBergeron, A.论文数: 0 引用数: 0 h-index: 0机构: Hop St Louis, Pulmonol, Paris, France Tauranga Hosp, Internal Med, Tauranga, New ZealandZeltser, D.论文数: 0 引用数: 0 h-index: 0机构: Tel Aviv Sourasky Med Ctr, Tel Aviv, Israel Tauranga Hosp, Internal Med, Tauranga, New ZealandMoudgil, H.论文数: 0 引用数: 0 h-index: 0机构: Princess Royal Hosp, Telford, Shrops, England Tauranga Hosp, Internal Med, Tauranga, New ZealandLimaye, A. P.论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Seattle, WA 98195 USA Tauranga Hosp, Internal Med, Tauranga, New ZealandCouturaud, F.论文数: 0 引用数: 0 h-index: 0机构: Ctr Hosp Reg & Univ Brest, Brest, France Tauranga Hosp, Internal Med, Tauranga, New ZealandNseir, W.论文数: 0 引用数: 0 h-index: 0机构: Nazareth EMMS Hosp, Nazareth, Israel Tauranga Hosp, Internal Med, Tauranga, New ZealandMcKevitt, M.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA USA Tauranga Hosp, Internal Med, Tauranga, New ZealandPorter, D.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA USA Tauranga Hosp, Internal Med, Tauranga, New ZealandJordan, R.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA USA Tauranga Hosp, Internal Med, Tauranga, New ZealandGuo, Y.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA USA Tauranga Hosp, Internal Med, Tauranga, New ZealandGerman, P.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA USA Tauranga Hosp, Internal Med, Tauranga, New ZealandWatkins, T. R.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA USA Tauranga Hosp, Internal Med, Tauranga, New ZealandGossage, D. L.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA USA Tauranga Hosp, Internal Med, Tauranga, New ZealandChien, J. W.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA USA Tauranga Hosp, Internal Med, Tauranga, New ZealandFalsey, A. R.论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Rochester, NY USA Tauranga Hosp, Internal Med, Tauranga, New Zealand
- [5] A Phase 2a Study Demonstrates That Gs-5806 Safely Reduces Viral Load And Clinical Illness In Healthy Adult Volunteers Infected With Respiratory Syncytial Virus (rsv)AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE, 2014, 189DeVincenzo, J.论文数: 0 引用数: 0 h-index: 0机构: Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USA论文数: 引用数: h-index:机构:Scaglioni, C.论文数: 0 引用数: 0 h-index: 0机构: Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USAHarrison, L.论文数: 0 引用数: 0 h-index: 0机构: Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USAMcBride, S.论文数: 0 引用数: 0 h-index: 0机构: Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USAMackman, R.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USAJordan, R.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USAXin, Y.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USARamanathan, S.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USAO'Riordan, T. G.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Seattle, WA USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USALewis, S.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Seattle, WA USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USAToback, S.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Seattle, WA USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USALin, S. -L.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USAChien, J.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Seattle, WA USA Univ Tennessee, Ctr Hlth Sci, Memphis, TN 38163 USA
- [6] GS-5806 Inhibits a Broad Range of Respiratory Syncytial Virus Clinical Isolates by Blocking the Virus-Cell Fusion ProcessANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2016, 60 (03) : 1264 - 1273Perron, Michel论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Gilead Sci, Foster City, CA USAStray, Kirsten论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Gilead Sci, Foster City, CA USAKinkade, April论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Gilead Sci, Foster City, CA USATheodore, Dorothy论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Gilead Sci, Foster City, CA USALee, Gary论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Gilead Sci, Foster City, CA USAEisenberg, Eugene论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Gilead Sci, Foster City, CA USASangi, Michael论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Gilead Sci, Foster City, CA USAGilbert, Brian E.论文数: 0 引用数: 0 h-index: 0机构: Baylor Coll Med, Houston, TX 77030 USA Gilead Sci, Foster City, CA USAJordan, Robert论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Gilead Sci, Foster City, CA USAPiedra, Pedro A.论文数: 0 引用数: 0 h-index: 0机构: Baylor Coll Med, Houston, TX 77030 USA Gilead Sci, Foster City, CA USAToms, Geoffery L.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Gilead Sci, Foster City, CA USAMackman, Richard论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Gilead Sci, Foster City, CA USACihlar, Tomas论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Gilead Sci, Foster City, CA USA
- [7] GS-5806 Inhibits Pre- to Postfusion Conformational Changes of the Respiratory Syncytial Virus Fusion ProteinANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2015, 59 (11) : 7109 - 7112Samuel, Dharmaraj论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Gilead Sci Inc, Foster City, CA 94404 USAXing, Weimei论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Gilead Sci Inc, Foster City, CA 94404 USANiedziela-Majka, Anita论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Gilead Sci Inc, Foster City, CA 94404 USAWong, Jinny S.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Gladstone Inst, San Francisco, CA 94143 USA Gilead Sci Inc, Foster City, CA 94404 USAHung, Magdeleine论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Gilead Sci Inc, Foster City, CA 94404 USABrendza, Katherine M.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Gilead Sci Inc, Foster City, CA 94404 USAPerron, Michel论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Gilead Sci Inc, Foster City, CA 94404 USAJordan, Robert论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Gilead Sci Inc, Foster City, CA 94404 USASperandio, David论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Gilead Sci Inc, Foster City, CA 94404 USALiu, Xiaohong论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Gilead Sci Inc, Foster City, CA 94404 USAMackman, Richard论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Gilead Sci Inc, Foster City, CA 94404 USASakowicz, Roman论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci Inc, Foster City, CA 94404 USA Gilead Sci Inc, Foster City, CA 94404 USA
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