One-pot synthesis of (5-alkyl-1,2,4-oxadiazol-3-yl)benzoic acids

被引：2

作者：

Baikov, Sergei V. ^{[1
]}

Krasovskaya, Galina G. ^{[1
]}

Kolobov, Aleksei V. ^{[1
]}

Kofanov, Evgenii R. ^{[1
]}

机构：

[1] Yaroslavl State Tech Univ, Yaroslavl 150023, Russia

来源：

MENDELEEV COMMUNICATIONS | 2015年 / 25卷 / 02期

关键词：

DESIGN; AGONISTS;

D O I：

10.1016/j.mencom.2015.03.021

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Heterocyclization of toluic acid amidoximes with acetic or propionic anhydrides affords 5-alkyl-3-tolyl-1,2,4-oxadiazoles, whose air oxidation in the same vessel gives (5-alkyl-1,2,4-oxadiazol-3-yl)benzoic acids.

引用

页码：138 / 139

页数：2

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