A VERSATILE SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF 3-OXO-2-ARYL-4-m-CHLOROPHENYL-5-TETRA-O-ACETYL-β-D-GLUCOPYRANOSYLIMINO-1,2,4-THIADIAZOLIDINES

被引：0
|
作者：
Bokade, Raksha S. [1 ]
Korpe, Gajanan V. [1 ]
机构：
[1] Sri Shivaji Coll, PG Dept Chem, Akola 444003, Maharashtra, India
来源：
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY | 2015年 / 24卷 / 03期
关键词：
PURINE NUCLEOSIDE ANALOGS; GLYCOGEN-PHOSPHORYLASE; HEPATITIS-B; INHIBITORS; AGENTS;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
3-Oxo-2-aryl-4-m-chloropheny1-5-tetra-O-acetyl-beta-D-glucopyranosylimino-1,2,4-thiadiazolidines have been prepared by the interaction of 1-aryl-3-m-chloro carbamide and tetra-O-acetyl-beta-D-glucopyranosyl-S-chloro-isothiocarbamoyl chloride. The identities of these newly synthesized compounds are established on the basis of elemental analysis IR, H-1 NMR, C-13 NMR, and mass spectral analysis. These compounds were assayed for their antibacterial and antifungal activity against E. coli, S. aureus, B. cereus, P. aeruginosa, P. vulgaris, A. niger and C. albicans to get potent bioactive molecule.
引用
收藏
页码：283 / 288
页数：6
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