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- [31] GSK973 Is an Inhibitor of the Second Bromodomains (BD2s) of the Bromodomain and Extra-Terminal (BET) FamilyACS MEDICINAL CHEMISTRY LETTERS, 2020, 11 (08): : 1581 - 1587Preston, Alex论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandAtkinson, Stephen J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandBamborough, Paul论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Platform Technol & Sci, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandChung, Chun-wa论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Platform Technol & Sci, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandGordon, Laurie J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Platform Technol & Sci, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandGrandi, Paola论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, D-69117 Heidelberg, Germany GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandGray, James R. J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandHarrison, Lee A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandLewis, Antonia J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Platform Technol & Sci, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandLugo, David论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandMessenger, Cassie论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Platform Technol & Sci, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandMichon, Anne-Marie论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, D-69117 Heidelberg, Germany GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandMitchell, Darren J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandPrinjha, Rab K.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandRioja, Inmaculada论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandSeal, Jon论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandTaylor, Simon论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandThesmar, Pierre论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandWall, Ian D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Platform Technol & Sci, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandWatson, J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandWoolven, James M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Platform Technol & Sci, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandDemont, Emmanuel H.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England
- [32] Identification of a Benzoisoxazoloazepine Inhibitor (CPI-0610) of the Bromodomain and Extra-Terminal (BET) Family as a Candidate for Human Clinical TrialsJOURNAL OF MEDICINAL CHEMISTRY, 2016, 59 (04) : 1330 - 1339Albrecht, Brian K.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Third Rock Ventures, 29 Newbury St 301, Boston, MA 02116 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USAGehling, Victor S.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USAHewitt, Michael C.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USAVaswani, Rishi G.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USACote, Alexandre论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USALeblanc, Yves论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Paraza Pharma Inc, 7171 Frederick Banting, Montreal, PQ H4S 1Z9, Canada Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USANasveschuk, Christopher G.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Broad Inst, 415 Main St, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USABellon, Steve论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USABergeron, Louise论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Bergeron Drug Discovery, Rome, Italy Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USACampbell, Robert论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Blueprint Med, 38 Sidney St 200, Cambridge, MA 02139 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USACantone, Nico论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USACooper, Michael R.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USACummings, Richard T.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USAJayaram, Hariharan论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Editas Med, 300 Third St, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USAJoshi, Shivangi论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Editas Med, 300 Third St, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USAMertz, Jennifer A.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USANeiss, Adrianne论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Huntsman Canc Inst, 2000 Circle Hope Dr, Salt Lake City, UT 84112 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USANormant, Emmanuel论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Surface Oncol, 215 First St,Suite 400-S, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USAO'Meara, Michael论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USAPardo, Eneida论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Forma Therapeut, 500 Arsenal St, Watertown, MA 02472 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USAPoy, Florence论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USASandy, Peter论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Evelo Therapeut, 620 Mem Dr,Suite 200 West, Cambridge, MA 02139 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USASupko, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Massachusetts Gen Hosp, Dana Farber Harvard Canc Ctr, 55 Fruit St,GRJ1025, Boston, MA 02114 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USASims, Robert J., III论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USAHarmange, Jean-Christophe论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Third Rock Ventures, 29 Newbury St 301, Boston, MA 02116 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USATaylor, Alexander M.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USAAudia, James E.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA
- [33] Targeting STAT5 in Hematologic Malignancies through Inhibition of the Bromodomain and Extra-Terminal (BET) Bromodomain Protein BRD2MOLECULAR CANCER THERAPEUTICS, 2014, 13 (05) : 1194 - 1205Liu, Suhu论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Univ, Sch Med, Boston, MA USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAWalker, Sarah R.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Univ, Sch Med, Boston, MA USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USANelson, Erik A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Univ, Sch Med, Boston, MA USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USACerulli, Robert论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Univ, Sch Med, Boston, MA USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA论文数: 引用数: h-index:机构:Toniolo, Patricia A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Univ, Sch Med, Boston, MA USA Univ Sao Paulo, Inst Biomed Sci, Dept Immunol, Sao Paulo, Brazil Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAQi, Jun论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Univ, Sch Med, Boston, MA USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAStone, Richard M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Univ, Sch Med, Boston, MA USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAWadleigh, Martha论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Univ, Sch Med, Boston, MA USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USABradner, James E.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Univ, Sch Med, Boston, MA USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAFrank, David A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Univ, Sch Med, Boston, MA USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA
- [34] BET protein inhibitor apabetalone (RVX-208) suppresses pro-inflammatory hyper-activation of monocytes from patients with cardiovascular disease and type 2 diabetesCLINICAL EPIGENETICS, 2020, 12 (01)Wasiak, Sylwia论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaDzobo, Kim E.论文数: 0 引用数: 0 h-index: 0机构: Univ Amsterdam, Amsterdam UMC, Amsterdam Cardiovasc Sci, Dept Expt Vasc Med, Meibergdreef 9, Amsterdam, Netherlands Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaRakai, Brooke D.论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaKaiser, Yannick论文数: 0 引用数: 0 h-index: 0机构: Univ Amsterdam, Amsterdam UMC, Amsterdam Cardiovasc Sci, Dept Vasc Med, Meibergdreef 9, Amsterdam, Netherlands Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaVersloot, Miranda论文数: 0 引用数: 0 h-index: 0机构: Univ Amsterdam, Amsterdam UMC, Amsterdam Cardiovasc Sci, Dept Expt Vasc Med, Meibergdreef 9, Amsterdam, Netherlands Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaBahjat, Mahnoush论文数: 0 引用数: 0 h-index: 0机构: Univ Amsterdam, Amsterdam UMC, Amsterdam Cardiovasc Sci, Dept Expt Vasc Med, Meibergdreef 9, Amsterdam, Netherlands Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaStotz, Stephanie C.论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaFu, Li论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaSweeney, Michael论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaJohansson, Jan O.论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaWong, Norman C. W.论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaStroes, Erik S. G.论文数: 0 引用数: 0 h-index: 0机构: Univ Amsterdam, Amsterdam UMC, Amsterdam Cardiovasc Sci, Dept Vasc Med, Meibergdreef 9, Amsterdam, Netherlands Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaKroon, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Univ Amsterdam, Amsterdam UMC, Amsterdam Cardiovasc Sci, Dept Expt Vasc Med, Meibergdreef 9, Amsterdam, Netherlands Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaKulikowski, Ewelina论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, 300-4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada
- [35] BET protein inhibitor apabetalone (RVX-208) suppresses pro-inflammatory hyper-activation of monocytes from patients with cardiovascular disease and type 2 diabetesClinical Epigenetics, 2020, 12Sylwia Wasiak论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCKim E. Dzobo论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCBrooke D. Rakai论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCYannick Kaiser论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCMiranda Versloot论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCMahnoush Bahjat论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCStephanie C. Stotz论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCLi Fu论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCMichael Sweeney论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCJan O. Johansson论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCNorman C. W. Wong论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCErik S. G. Stroes论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCJeffrey Kroon论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMCEwelina Kulikowski论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp,Department of Experimental Vascular Medicine, Amsterdam Cardiovascular Sciences, Amsterdam UMC
- [36] Bromodomain Inhibitor Review: Bromodomain and Extra-terminal Family Protein Inhibitors as a Potential New Therapy in Central Nervous System TumorsCUREUS, 2016, 8 (05):Wadhwa, Elizabeth论文数: 0 引用数: 0 h-index: 0机构: UCSF, Pediat, San Francisco, CA 94143 USA UCSF, Pediat, San Francisco, CA 94143 USANicolaides, Theodore论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Neurol Surg & Pediat, San Francisco, CA 94143 USA UCSF, Pediat, San Francisco, CA 94143 USA
- [37] Deacetylase inhibitors repress STAT5-mediated transcription by interfering with bromodomain and extra-terminal (BET) protein functionNUCLEIC ACIDS RESEARCH, 2015, 43 (07) : 3524 - 3545Pinz, Sophia论文数: 0 引用数: 0 h-index: 0机构: Univ Regensburg, Inst Immunol, Signaling Res Grp Stat5, D-93053 Regensburg, Germany Univ Regensburg, Inst Immunol, Signaling Res Grp Stat5, D-93053 Regensburg, GermanyUnser, Samy论文数: 0 引用数: 0 h-index: 0机构: Univ Regensburg, Inst Immunol, Signaling Res Grp Stat5, D-93053 Regensburg, Germany Univ Regensburg, Inst Immunol, Signaling Res Grp Stat5, D-93053 Regensburg, GermanyBuob, Dominik论文数: 0 引用数: 0 h-index: 0机构: Univ Regensburg, Inst Immunol, Signaling Res Grp Stat5, D-93053 Regensburg, Germany Univ Regensburg, Inst Immunol, Signaling Res Grp Stat5, D-93053 Regensburg, GermanyFischer, Philipp论文数: 0 引用数: 0 h-index: 0机构: Univ Regensburg, Inst Immunol, Signaling Res Grp Stat5, D-93053 Regensburg, Germany Univ Regensburg, Inst Immunol, Signaling Res Grp Stat5, D-93053 Regensburg, GermanyJobst, Belinda论文数: 0 引用数: 0 h-index: 0机构: Univ Regensburg, Inst Immunol, Signaling Res Grp Stat5, D-93053 Regensburg, Germany Univ Regensburg, Inst Immunol, Signaling Res Grp Stat5, D-93053 Regensburg, Germany论文数: 引用数: h-index:机构:
- [38] RVX-208, a BET-inhibitor for treating atherosclerotic cardiovascular disease, raises ApoA-I/HDL and represses pathways that contribute to cardiovascular disease (vol 247, pg 48, 2016)ATHEROSCLEROSIS, 2016, 253 : 345 - 345Gilham, Dean论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaWasiak, Sylwia论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaTsujikawa, Laura M.论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaHalliday, Christopher论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaNorek, Karen论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaPatel, Reena G.论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaKulikowski, Ewelina论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaJohansson, Jan论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, San Francisco, CA USA Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaSweeney, Michael论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, San Francisco, CA USA Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, CanadaWong, Norman C. W.论文数: 0 引用数: 0 h-index: 0机构: Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada Resverlogix Corp, Suite 300,4820 Richard Rd SW, Calgary, AB T3E 6L1, Canada
- [39] Structure-Based Discovery and Development of a Series of Potent and Selective Bromodomain and Extra-Terminal Protein InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2019, 62 (18) : 8642 - 8663Hu, Jianping论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Materia Med, State Key Lab Drug Res, Dept Med Chem, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Materia Med, State Key Lab Drug Res, Dept Med Chem, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R ChinaTian, Chang-Qing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Materia Med, State Key Lab Drug Res, Div Antitumor Pharmacol, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Materia Med, State Key Lab Drug Res, Dept Med Chem, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R ChinaDamaneh, Mohammadali 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