Studies on the synthesis and reactivity of novel benzofuran-2-yl-[3-methyl-3-phenylcyclobutyl] methanones and their antimicrobial activity

被引:15
作者
Koca, M
Ahmedzade, M
Cukurovali, A [1 ]
Kazaz, C
机构
[1] Firat Univ, Fac Arts & Sci, Dept Chem, TR-23119 Elazig, Turkey
[2] Ataturk Univ, Fac Arts & Scu, Dept Chem, Erzurum, Turkey
关键词
furans; cyclobutane; oxime; thiazole; thiosemicarbazone;
D O I
10.3390/10070747
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
Preparation in excellent yields of cyclobutyl benzofuran-2-yl- and naphthofuran-2-yl-ketones, the corresponding ketoximes and thiosemicarbazones, ether derivatives of the ketoximes and thiazoles derived from the thiosernicarbazones are described. Two of the synthesized compounds have been tested against eight different microorganisms and found to be active against some of the species studied.
引用
收藏
页码:747 / 754
页数:8
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