Potent dual 5-lipoxygenase inhibitor and PAF receptor antagonist

被引:0
|
作者
Lloyd, AW [1 ]
机构
[1] Univ Brighton, Dept Pharm, Brighton BN2 4GJ, E Sussex, England
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:424 / 424
页数:1
相关论文
共 50 条
  • [1] Anti-inflammatory activities of LDP-392, a dual PAF receptor antagonist and 5-lipoxygenase inhibitor
    Qian, CG
    Hwang, SB
    Libertine-Garahan, L
    Eckman, JB
    Cai, X
    Scannell, RT
    Yeh, CG
    PHARMACOLOGICAL RESEARCH, 2001, 44 (03) : 213 - 220
  • [2] CMI-206 - A POTENT DUAL PLATELET-ACTIVATING-FACTOR ANTAGONIST AND 5-LIPOXYGENASE INHIBITOR
    HUSSOIN, MS
    CAI, X
    SCANNELL, RT
    YAEGER, D
    KILLIAN, DB
    ECKMAN, J
    HWANG, SB
    LIBERTINEGARAHAN, L
    QIAN, CG
    YEH, CG
    IP, S
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1995, 5 (06) : 643 - 648
  • [3] Discovery of ucb 35440: A potent and orally active dual acting 5-lipoxygenase inhibitor and H1 receptor antagonist.
    Cai, X
    Arrington, M
    Bayless, L
    Eckman, J
    Eckert, M
    Ene, D
    Ellis, J
    Hussoin, S
    Latham, M
    Lewis, T
    Libertine, L
    Nicolas, JM
    Scannell, R
    Selig, W
    Schwartz, E
    Wels, B
    Wypij, D
    Young, M
    Zou, D
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2002, 224 : U62 - U62
  • [4] A FLAVONOID, NEW POTENT 5-LIPOXYGENASE INHIBITOR
    KOHNO, SW
    TAIRA, M
    OHATA, K
    YAMAMOTO, S
    YOKOYAMA, C
    HORIE, T
    ANNALS OF ALLERGY, 1985, 55 (02): : 362 - 362
  • [5] DIPYRIDAMOLE - A POTENT AND SPECIFIC 5-LIPOXYGENASE INHIBITOR
    CARTER, GW
    DYER, R
    YOUNG, P
    FEDERATION PROCEEDINGS, 1985, 44 (04) : 904 - 904
  • [6] In vitro characterization of dual action 5-lipoxygenase inhibitor/H1 receptor antagonist compounds
    Wypij, D
    Cai, X
    Eckert, M
    Eckman, J
    Ellis, J
    Hussoin, S
    Lewis, T
    Scannell, R
    Selig, W
    Wels, B
    Wenberg, K
    Young, M
    MOLECULAR BIOLOGY OF THE CELL, 2002, 13 : 401A - 401A
  • [7] Antiallergic effect of ardisiaquinone A, a potent 5-lipoxygenase inhibitor
    Fukuishi, N
    Takada, T
    Fukuyama, Y
    Akagi, M
    PHYTOMEDICINE, 2001, 8 (06) : 460 - 464
  • [8] DISULFIRAM IS A POTENT INHIBITOR OF RAT 5-LIPOXYGENASE ACTIVITY
    CHOO, LY
    RIENDEAU, D
    CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1987, 65 (12) : 2503 - 2506
  • [9] Synthesis and Structural Proof of a Potent 5-Lipoxygenase Inhibitor
    Balu, Devipriya
    Poomani, Kumaradhas
    Nagabushanam, Kalyanam
    Balasubramanium, Sridhar
    Ramanujam, Rajendran
    Muhammed, Majeed
    JOURNAL OF CHEMICAL CRYSTALLOGRAPHY, 2011, 41 (05) : 697 - 702
  • [10] Synthesis and Structural Proof of a Potent 5-Lipoxygenase Inhibitor
    Devipriya Balu
    Kumaradhas Poomani
    Kalyanam Nagabushanam
    Sridhar Balasubramanium
    Rajendran Ramanujam
    Majeed Muhammed
    Journal of Chemical Crystallography, 2011, 41 : 697 - 702