Development and utilization of cultured human mast cells for high throughput small molecule drug discovery

被引:0
作者
Rossi, A
Holland, S
Woronicz, J
Quast, J
Argade, A
Sylvain, C
Juencke, S
Sula, C
Tombo, W
Goodrich, B
Pine, P
Scheerens, H
Natarajan, G
Li, WB
Bennett, M
Daniel, R
Wagner, G
Singh, R
Molineaux, S
Payan, D
机构
[1] Rigel Pharmaceut Inc, Cell Biol, San Francisco, CA 94080 USA
[2] Rigel Pharmaceut Inc, Chem, San Francisco, CA 94080 USA
[3] Rigel Pharmaceut Inc, High Throughput Screening, San Francisco, CA 94080 USA
[4] Rigel Pharmaceut Inc, Pharmacol, San Francisco, CA 94080 USA
[5] Rigel Pharmaceut Inc, Chief Sci Off, San Francisco, CA 94080 USA
关键词
D O I
暂无
中图分类号
Q2 [细胞生物学];
学科分类号
071009 ; 090102 ;
摘要
2824
引用
收藏
页码:512A / 513A
页数:2
相关论文
共 50 条
[21]   Development of a Zebrafish Sepsis Model for High-Throughput Drug Discovery [J].
Philip, Anju M. ;
Wang, Youdong ;
Mauro, Antonio ;
El-Rass, Suzan ;
Marshall, John C. ;
Lee, Warren L. ;
Slutsky, Arthur S. ;
dos Santos, Claudia C. ;
Wen, Xiao-Yan .
MOLECULAR MEDICINE, 2017, 23 :134-148
[22]   Notes on AEMS methods development for high throughput experimentation in drug discovery [J].
Verma, Meghav ;
Hoxie, Nate ;
Janiszewski, John ;
Bonney, Charles ;
Hall, Matthew D. ;
Michael, Sam ;
Covey, Tom ;
Shrimp, Jonathan H. .
SLAS TECHNOLOGY, 2024, 29 (06)
[23]   High-throughput discovery of novel small-molecule inhibitors of acid Ceramidase [J].
Aseeri, Mazen ;
Abad, Jose Luis ;
Delgado, Antonio ;
Fabrias, Gemma ;
Triola, Gemma ;
Casas, Josefina .
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2023, 38 (01) :343-348
[24]   High Throughput Screening for Small Molecule Enhancers of the Interferon Signaling Pathway to Drive Next-Generation Antiviral Drug Discovery [J].
Patel, Dhara A. ;
Patel, Anand C. ;
Nolan, William C. ;
Zhang, Yong ;
Holtzman, Michael J. .
PLOS ONE, 2012, 7 (05)
[25]   Leveraging Superficially Porous Particle Technology to Develop High-Throughput HPLC Methods for Small-Molecule Drug Discovery [J].
Nancharaiah Tellakula ;
Mallikarjuna Guna ;
Mitalee Das ;
Vaishali Bane ;
Siddheshwar Kisan Chauthe ;
Arvind Mathur ;
Muralidhararao Bagadi ;
Khemraj Bairwa ;
Amrita Roy .
Chromatographia, 2023, 86 :437-446
[26]   Leveraging Superficially Porous Particle Technology to Develop High-Throughput HPLC Methods for Small-Molecule Drug Discovery [J].
Tellakula, Nancharaiah ;
Guna, Mallikarjuna ;
Das, Mitalee ;
Bane, Vaishali ;
Chauthe, Siddheshwar Kisan ;
Mathur, Arvind ;
Bagadi, Muralidhararao ;
Bairwa, Khemraj ;
Roy, Amrita .
CHROMATOGRAPHIA, 2023, 86 (06) :437-446
[27]   Small Molecule Crystal Structures in Drug Discovery [J].
Groom, Colin .
MULTIFACETED ROLES OF CRYSTALLOGRAPHY IN MODERN DRUG DISCOVERY, 2015, :107-114
[28]   DRUG DISCOVERY Small molecule targets RNA [J].
Satyanarayana, Megha .
CHEMICAL & ENGINEERING NEWS, 2021, 99 (31) :8-8
[29]   Igniting Small-Molecule Drug Discovery [J].
Steinhagen, Henning .
CHEMMEDCHEM, 2016, 11 (02) :148-149
[30]   Small Molecule Drug Discovery for Pediatric Diseases [J].
Trippier, Paul C. .
MINI-REVIEWS IN MEDICINAL CHEMISTRY, 2016, 16 (06) :428-429