COPPER-CATALYZED DOMINO REACTION OF HETEROALLENES TOWARDS BENZO-HETEROCYCLE COMPOUNDS

被引:8
作者
Wang, Fei [1 ]
Zhao, Peng [1 ]
Xi, Chanjuan [1 ]
机构
[1] Tsinghua Univ, Dept Chem, Key Lab Bioorgan Phosphorus Chem & Chem Biol, Minist Educ, Beijing 100084, Peoples R China
基金
中国国家自然科学基金;
关键词
Carbodiimide; Isothiocyanate; Carbon Disulfide; Domino Reaction; Benzo-Heterocycle; ONE-POT SYNTHESIS; BENZIMIDAZOLE DERIVATIVES; O-HALOANILINES; TANDEM REACTION; SMALL-MOLECULE; INHIBITORS; EFFICIENT; 2(3H)-BENZOTHIAZOLETHIONES; 2-AMINOBENZIMIDAZOLES; ISOTHIOCYANATES;
D O I
10.3987/REV-11-SR(P)6
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The present review summarizes information on the copper-catalyzed reaction of heteroallenes, including carbodiimides, isothiocyanates, and carbon disulfide, with o-halobenzenamines or o-halophenols or o-halobenzamides for constructing benzo-heterocycle compounds via domino nucleophilic addition/cyclization reactions.
引用
收藏
页码:209 / 221
页数:13
相关论文
共 56 条
[1]   Synthesis and pharmacological evaluation of 3-cyclohexyl-2-substituted hydrazino-3H-quinazolin-4-ones as analgesic and anti-inflammatory agents [J].
Alagarsamy, Veerachamy ;
Shankar, Durairaj ;
Solomon, Viswas Raja ;
Sheorey, Rajendra Vasant ;
Parthiban, Periyasamy .
ACTA PHARMACEUTICA, 2009, 59 (01) :75-88
[2]  
[Anonymous], 1998, INDIAN DRUGS
[3]   Synthesis of 1H-quinazoline-4-ones using intramolecular aromatic nucleophilic substitution [J].
Bowman, WR ;
Heaney, H ;
Smith, PHG .
ARKIVOC, 2003, :434-442
[4]   An intramolecular palladium-catalysed aryl amination reaction to produce benzimidazoles [J].
Brain, CT ;
Brunton, SA .
TETRAHEDRON LETTERS, 2002, 43 (10) :1893-1895
[5]   2-Ethoxybenzoxazole as a bioisosteric replacement of an ethyl benzoate group in a human rhinovirus (HRV) capsid binder [J].
Brown, RN ;
Cameron, R ;
Chalmers, DK ;
Hamilton, S ;
Luttick, A ;
Krippner, GY ;
McConnell, DB ;
Nearn, R ;
Stanislawski, PC ;
Tucker, SP ;
Watson, KG .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2005, 15 (08) :2051-2055
[6]   Transition-Metal-Free O-, S-, and N-Arylation of Alcohols, Thiols, Amides, Amines, and Related Heterocycles [J].
Cano, Rafael ;
Ramon, Diego J. ;
Yus, Miguel .
JOURNAL OF ORGANIC CHEMISTRY, 2011, 76 (02) :654-660
[7]   STRUCTURE OF A23187, A DIVALENT-CATION IONOPHORE [J].
CHANEY, MO ;
DEMARCO, PV ;
JONES, ND ;
OCCOLOWI.JL .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1974, 96 (06) :1932-1933
[8]   Convenient strategies for the preparation of modified 2(3H)-benzothiazolethiones [J].
Chaudhuri, NC .
SYNTHETIC COMMUNICATIONS, 1996, 26 (20) :3783-3790
[9]   The first low μM SecA inhibitors [J].
Chen, Weixuan ;
Huang, Ying-ju ;
Gundala, Sushma Reddy ;
Yang, Hsiuchin ;
Li, Minyong ;
Tai, Phang C. ;
Wang, Binghe .
BIOORGANIC & MEDICINAL CHEMISTRY, 2010, 18 (04) :1617-1625
[10]   Synthesis of 2-Aminobenzothiazole via Copper(I)-Catalyzed Tandem Reaction of 2-Iodobenzenamine with Isothiocyanate [J].
Ding, Qiuping ;
He, Xiaodan ;
Wu, Jie .
JOURNAL OF COMBINATORIAL CHEMISTRY, 2009, 11 (04) :587-591