Prostaglandin D2 receptor antagonism: a novel therapeutic option for eosinophilic asthma?

被引:7
作者
Brusselle, Guy G. [1 ,2 ,3 ]
Provoost, Sharen [1 ]
Maes, Tania [1 ]
机构
[1] Ghent Univ Hosp, Dept Resp Med, B-9000 Ghent, Belgium
[2] Erasmus MC, Dept Epidemiol, Rotterdam, Netherlands
[3] Erasmus MC, Dept Resp Med, Rotterdam, Netherlands
关键词
CRTH2; ANTAGONIST; INFLAMMATION;
D O I
10.1016/S2213-2600(16)30201-6
中图分类号
R4 [临床医学];
学科分类号
1002 ; 100602 ;
摘要
引用
收藏
页码:676 / 677
页数:2
相关论文
共 50 条
  • [21] The Roles of Type 2 Cytotoxic T Cells in Inflammation, Tissue Remodeling, and Prostaglandin (PG) D2 Production Are Attenuated by PGD2 Receptor 2 Antagonism
    Chen, Wentao
    Luo, Jian
    Ye, Yuan
    Hoyle, Ryan
    Liu, Wei
    Borst, Rowie
    Kazani, Shamsah
    Shikatani, Eric A.
    Erpenbeck, Veit J.
    Pavord, Ian D.
    Klenerman, Paul
    Sandham, David A.
    Xue, Luzheng
    JOURNAL OF IMMUNOLOGY, 2021, 206 (11) : 2714 - 2724
  • [22] Prostaglandin D2 as a mediator of lymphopenia and a therapeutic target in COVID-19 disease
    Gupta, Ajay
    Chiang, Kate Chander
    MEDICAL HYPOTHESES, 2020, 143
  • [23] Development of a prostaglandin D2 receptor antagonist:: discovery of a new chemical lead
    Torisu, K
    Kobayashi, K
    Iwahashi, M
    Egashira, H
    Nakai, Y
    Okada, Y
    Nanbu, F
    Ohuchida, S
    Nakai, H
    Toda, M
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2005, 40 (05) : 505 - 519
  • [24] Prostaglandin D2 regulates human colonic ion transport via the DP1 receptor
    Medani, M.
    Collins, D.
    Mohan, H. M.
    Walsh, E.
    Winter, D. C.
    Baird, A. W.
    LIFE SCIENCES, 2015, 122 : 87 - 91
  • [25] Ramatroban (BAY u 3405):: A novel dual antagonist of TXA2 receptor and CRTh2, a newly identified prostaglandin D2 receptor
    Ishizuka, T
    Matsui, T
    Okamoto, Y
    Ohta, A
    Shichijo, M
    CARDIOVASCULAR DRUG REVIEWS, 2004, 22 (02): : 71 - 90
  • [26] Attenuation of Laser-Induced Choroidal Neovascularization by Blockade of Prostaglandin D2 Receptor 2
    Soga, Hirotsugu
    Inoue, Tatsuya
    Urade, Yoshihiro
    Ueta, Takashi
    Kawashima, Hidetoshi
    Kaburaki, Toshikatsu
    Aihara, Makoto
    TRANSLATIONAL VISION SCIENCE & TECHNOLOGY, 2023, 12 (05):
  • [27] Prostaglandin D2 sustains the pyrogenic effect of prostaglandin E2
    Gao, Wei
    Schmidtko, Achim
    Lu, Ruirui
    Brenneis, Christian
    Angioni, Carlo
    Schmidt, Ronald
    Geisslinger, Gerd
    EUROPEAN JOURNAL OF PHARMACOLOGY, 2009, 608 (1-3) : 28 - 31
  • [28] Safety and efficacy of the prostaglandin D2 receptor antagonist AMG 853 in asthmatic patients
    Busse, William W.
    Wenzel, Sally E.
    Meltzer, Eli O.
    Kerwin, Edward M.
    Liu, Mark C.
    Zhang, Nan
    Chon, Yun
    Budelsky, Alison L.
    Lin, Joseph
    Lin, Shao-Lee
    JOURNAL OF ALLERGY AND CLINICAL IMMUNOLOGY, 2013, 131 (02) : 339 - 345
  • [29] The effect of MK-0524, a prostaglandin D2 receptor antagonist, on prostaglandin D2-induced nasal airway obstruction in healthy volunteers
    Van Hecken, A.
    Depre, M.
    De Lepeleire, I.
    Thach, C.
    Oeyen, M.
    Van Effen, J.
    Laethem, T.
    Mazina, K.
    Crumley, T.
    Wenning, L.
    Gottesdiener, K. M.
    Deutsch, P.
    Clement, P.
    Lai, E.
    de Hoon, J. N.
    EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 2007, 63 (02) : 135 - 141
  • [30] CRTH2, a prostaglandin D2 receptor, mediates depression-related behavior in mice
    Onaka, Yusuke
    Shintani, Norihito
    Nakazawa, Takanobu
    Haba, Ryota
    Ago, Yukio
    Wang, Hyper
    Kanoh, Takuya
    Hayata-Takano, Atsuko
    Hirai, Hiroyuki
    Nagata, Kin-ya
    Nakamura, Masataka
    Hashimoto, Ryota
    Matsuda, Toshio
    Waschek, James A.
    Kasai, Atsushi
    Nagayasu, Kazuki
    Baba, Akemichi
    Hashimoto, Hitoshi
    BEHAVIOURAL BRAIN RESEARCH, 2015, 284 : 131 - 137