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BMS-986165 IS A HIGHLY POTENT AND SELECTIVE ALLOSTERIC INHIBITOR OF TYK2, BLOCKS IL-12, IL-23 AND TYPE I INTERFERON SIGNALING AND PROVIDES FOR ROBUST EFFICACY IN PRECLINICAL MODELS OF INFLAMMATORY BOWEL DISEASE
被引:0
|
作者
:
Xie, Jenny H.
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0
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0
h-index:
0
Xie, Jenny H.
Gillooly, Kathleen
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0
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0
h-index:
0
Gillooly, Kathleen
Zhang, Yifan
论文数:
0
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0
h-index:
0
Zhang, Yifan
Yang, Xiaoxia
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0
引用数:
0
h-index:
0
Yang, Xiaoxia
Zupa-Fernandez, Adriana
论文数:
0
引用数:
0
h-index:
0
Zupa-Fernandez, Adriana
Cheng, Lihong
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0
引用数:
0
h-index:
0
Cheng, Lihong
Strnad, Joann
论文数:
0
引用数:
0
h-index:
0
Strnad, Joann
Heimrich, Elizabeth
论文数:
0
引用数:
0
h-index:
0
Heimrich, Elizabeth
Zhou, Xiaodi
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0
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0
h-index:
0
Zhou, Xiaodi
Chen, Jing
论文数:
0
引用数:
0
h-index:
0
Chen, Jing
Chaudhry, Charu
论文数:
0
引用数:
0
h-index:
0
Chaudhry, Charu
Li, Sha
论文数:
0
引用数:
0
h-index:
0
Li, Sha
Moslin, Ryan
论文数:
0
引用数:
0
h-index:
0
Moslin, Ryan
Wrobleski, Stephen
论文数:
0
引用数:
0
h-index:
0
Wrobleski, Stephen
Burke, James
论文数:
0
引用数:
0
h-index:
0
Burke, James
机构
:
来源
:
GASTROENTEROLOGY
|
2018年
/ 154卷
/ 06期
关键词
:
D O I
:
暂无
中图分类号
:
R57 [消化系及腹部疾病];
学科分类号
:
摘要
:
349
引用
收藏
页码:S1357 / S1357
页数:1
相关论文
共 3 条
[1]
BMS-986165 Is a Highly Potent and Selective Allosteric Inhibitor of Tyk2, Blocks IL-12, IL-23 and Type I Interferon Signaling and Provides for Robust Efficacy in Preclinical Models of Systemic Lupus Erythematosus and Inflammatory Bowel Disease
Gillooly, Kathleen
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Gillooly, Kathleen
Zhang, Yifan
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0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Zhang, Yifan
Yang, Xiaoxia
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0
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0
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机构:
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Yang, Xiaoxia
Zupa-Fernandez, Adriana
论文数:
0
引用数:
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h-index:
0
机构:
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Zupa-Fernandez, Adriana
Cheng, Lihong
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Cheng, Lihong
Strnad, Joann
论文数:
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引用数:
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h-index:
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机构:
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Strnad, Joann
Cunningham, Mark
论文数:
0
引用数:
0
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0
机构:
Bristol Myers Squibb, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Cunningham, Mark
Heimrich, Elizabeth
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Heimrich, Elizabeth
Zhou, Xiadi
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Zhou, Xiadi
Chen, Jing
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Leads Discovery & Optimizat, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Chen, Jing
Chaudhry, Charu
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Leads Discovery & Optimizat, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Chaudhry, Charu
Li, Sha
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Leads Discovery & Optimizat, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Li, Sha
McIntyre, Kim
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
McIntyre, Kim
Carman, Julie
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Discovery Translat Sci Grp, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Carman, Julie
Moslin, Ryan
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Immunosci Discovery Chem, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Moslin, Ryan
Wrobleski, Stephen
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Immunosci Discovery Chem, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Wrobleski, Stephen
Weinstein, David
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Immunosci Discovery Chem, Princeton, NJ USA
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
Weinstein, David
Burke, James
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Immunosci Discovery Biol, Princeton, NJ USA
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Burke, James
ARTHRITIS & RHEUMATOLOGY,
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68
[2]
A selective TYK2 inhibitor, BMS-986165, decreases the transcriptional signature of Th17, IL-12, and interferon pathways in skin of psoriasis: results from a Phase 2 trial
Catlett, I.
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Princeton, NJ USA
Bristol Myers Squibb, Princeton, NJ USA
Catlett, I.
Hu, S.
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb, Princeton, NJ USA
Bristol Myers Squibb, Princeton, NJ USA
Hu, S.
Banerjee, S.
论文数:
0
引用数:
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h-index:
0
机构:
Bristol Myers Squibb, Princeton, NJ USA
Bristol Myers Squibb, Princeton, NJ USA
Banerjee, S.
Krueger, J. G.
论文数:
0
引用数:
0
h-index:
0
机构:
Rockefeller Univ, 1230 York Ave, New York, NY 10021 USA
Bristol Myers Squibb, Princeton, NJ USA
Krueger, J. G.
JOURNAL OF INVESTIGATIVE DERMATOLOGY,
2019,
139
(09)
: B2
-
B2
[3]
Selective Inhibition of Tyrosine Kinase 2 (TYK2) with BMS-986165 Is Efficacious in IL-23-Mediated Diseases: Evidence from Preclinical IBD Models and From a Psoriasis Study
Burke, James R.
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Bristol Myers Squibb, Princeton, NJ USA
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Xie, Jenny
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Bristol Myers Squibb, Princeton, NJ USA
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论文数:
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AMERICAN JOURNAL OF GASTROENTEROLOGY,
2018,
113
: S354
-
S354
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