Solid-phase synthesis of C-terminal peptide amides from N-tetrachlorophthaloyl protected amino acids

被引：5

作者：

Cros, E ^{[1
]}

Planas, M ^{[1
]}

Mejías, X ^{[1
]}

Bardají, E ^{[1
]}

机构：

[1] Univ Girona, Dept Chem, Girona 17071, Spain

来源：

TETRAHEDRON LETTERS | 2001年 / 42卷 / 35期

关键词：

D O I：

10.1016/S0040-4039(01)01193-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new strategy for solid-phase synthesis of C-terminal peptide amides based on the use of N-tetrachlorophthaloyl protected amino acids with acid-labile side-chain protection is described. (C) 2001 Elsevier Science Ltd. All rights reserved.

引用

页码：6105 / 6107

页数：3

共 50 条

[31] FACILE SYNTHESIS OF PROTECTED C-TERMINAL PEPTIDE SEGMENTS BY FMOC/BU(T) SOLID-PHASE PROCEDURES ON N-FMOC-9-AMINO-XANTHEN-3-YLOXYMETHYL POLYSTYRENE RESIN
CHAN, WC
WHITE, PD
BEYTHIEN, J
STEINAUER, R
JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1995, (05) : 589 - 592
[32] SEQUENTIAL POLYPEPTIDES - SYNTHESIS OF N-PROTECTED, C-ACTIVATED PEPTIDES FROM C-TERMINAL RESIDUES OF AMINO ACIDS
KAPOOR, A
GERENCSER, LW
JOURNAL OF PHARMACEUTICAL SCIENCES, 1969, 58 (08) : 976 - +
[33] Synthesis of amide N-H protected amino acids for use in solid phase peptide synthesis
Chapman, Ashley
Black, Sarah
Steinkruger, Jay D.
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248
[34] Solid phase synthesis of peptide C-terminal semicarbazones and aldehydes
Patterson, JA
Ramage, R
TETRAHEDRON LETTERS, 1999, 40 (33) : 6121 - 6124
[35] Arylboronate Ester Protected Amino Acids as Orthogonal Building Blocks for Fmoc Solid-Phase Peptide Synthesis
Liu, Chao
Zou, Yan
Song, Hui
Jiang, Yuan-Ye
Hu, Hong-Gang
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2017, 2017 (39) : 5916 - 5920
[36] Solid-phase synthesis of C-terminal peptide libraries for studying the specificity of enzymatic protein prenylation
Wang, Yen-Chih
Distefano, Mark D.
CHEMICAL COMMUNICATIONS, 2012, 48 (66) : 8228 - 8230
[37] Fmoc solid-phase synthesis of C-terminal peptide thioesters by formation of a pyroglutamyl imide moiety
Tofteng, A. Pernille
Conde-Frieboes, Kilian W.
Hoeg-Jensen, Thomas
Jensen, Knud J.
JOURNAL OF PEPTIDE SCIENCE, 2008, 14 (08) : 15 - 15
[38] Solid-Phase Peptide Synthesis - Evaluation of Resin Loading and Preparation of an Amide C-Terminal Dipeptide
Nicolau, Ioana
Paun, Anca
Popescu, Codruta C.
Hadade, Niculina D. D.
Matache, Mihaela
JOURNAL OF CHEMICAL EDUCATION, 2023, 100 (06) : 2430 - 2434
[39] A new Fmoc-compatible method for the solid-phase synthesis of peptide C-terminal α-thioesters
Camarero, JA
de Yoreo, J
Mitchell, AR
BIOPOLYMERS, 2003, 71 (03) : 363 - 363
[40] An alternate preparation of thioester resin linkers for solid-phase synthesis of peptide C-terminal thioacids
Goldstein, AS
Gelb, MH
TETRAHEDRON LETTERS, 2000, 41 (16) : 2797 - 2800

← 1 2 3 4 5 →