Click-tambjamines as efficient and tunable bioactive anion transporters

被引：18
作者：
Carreira-Barral, Israel [1 ]
Mielczarek, Marcin [1 ]
Alonso-Carrillo, Daniel [1 ]
Capurro, Valeria [2 ]
Soto-Cerrato, Vanessa [3 ]
Tomas, Ricardo Perez [3 ]
Caci, Emanuela [2 ]
Garcia-Valverde, Maria [1 ]
Quesada, Roberto [1 ]
机构：
[1] Univ Burgos, Dept Quim, Burgos 09001, Spain
[2] IRCSS Ist Giannina Gaslini, UOC Genet Med, Genoa, Italy
[3] Univ Barcelona, Dept Pathol & Expt Therapeut, Fac Med, Barcelona, Spain
来源：
CHEMICAL COMMUNICATIONS | 2020年 / 56卷 / 21期
基金：
欧盟地平线“2020”;
关键词：
RECEPTOR;
D O I：
10.1039/d0cc00643b
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A novel class of transmembrane anion carriers, the click-tambjamines, display remarkable anionophoric activities in model liposomes and living cells. The versatility of this building block for the generation of molecular diversity offers promise to develop future drugs based on this design.
引用
收藏
页码：3218 / 3221
页数：4
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