Azide-Free Synthesis of 1,2,3-Triazoles: New Opportunity for Sustainable Synthesis

被引：47

作者：

Wan, Jie-Ping ^{[1
,2
]}

Hu, Deqing ^{[1
]}

Liu, Yunyun ^{[1
,2
]}

Sheng, Shouri ^{[1
,2
]}

机构：

[1] Jiangxi Normal Univ, Coll Chem & Chem Engn, Nanchang 330022, Peoples R China

[2] Jiangxi Normal Univ, Key Lab Funct Small Organ Mol, Minist Educ, Nanchang 330022, Peoples R China

来源：

CHEMCATCHEM | 2015年 / 7卷 / 06期

关键词：

1,2,3-triazole; azide-free; click chemistry; diversity; sustainability; METAL-FREE SYNTHESIS; ALKYNE CYCLOADDITION; N-TOSYLHYDRAZONES; 1.3-DIPOLARE CYCLOADDITIONEN; 1,3-DIPOLAR CYCLOADDITION; REGIOSELECTIVE SYNTHESIS; TRIAZOLE FORMATION; HIV-1; PROTEASE; COPPER-FREE; HUISGEN;

D O I：

10.1002/cctc.201500001

中图分类号：

O64 [物理化学（理论化学）、化学物理学];

学科分类号：

070304 ; 081704 ;

摘要：

A bright future for triazoles: The recent breakthrough in the synthesis of 1,2,3-triazoles is highlighted for its significance as a new tool in the chemistry of 1,2,3-triazoles following the classical CuAAC and metal-free protocols. © 2015 WILEY-VCH Verlag GmbH & Co. KGaA, Weinheim.

引用

页码：901 / 903

页数：3

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