Syntheses and optimization of new GS39783 analogues as positive allosteric modulators of GABAB receptors

被引：51

作者：

Guery, Sebastien ^{[1
]}

Floersheim, Philipp ^{[1
]}

Kaupmann, Klemens ^{[1
]}

Froestl, Wolfgang ^{[1
]}

机构：

[1] Novartis Inst Biomed Res, Neurosci, Novartis Pharma, CH-4002 Basel, Switzerland

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 2007年 / 17卷 / 22期

关键词：

GABA(B) positive allosteric modulators; GS39783; drug addiction;

D O I：

10.1016/j.bmcl.2007.09.023

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：6206 / 6211

页数：6

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