High throughput screening for inhibition of cytochrome p450 metabolism

被引:0
作者
Crespi, CL [1 ]
Miller, VP [1 ]
Penman, BW [1 ]
机构
[1] GENTEST Corp, Woburn, MA 01801 USA
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D O I
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中图分类号
R914 [药物化学];
学科分类号
100701 ;
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页码:457 / 471
页数:15
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共 16 条
[1]  
BURKE MD, 1983, CHEM-BIOL INTERACT, V45, P243
[2]   CHARACTERIZATION OF THE INHIBITION OF P4501A2 BY FURAFYLLINE [J].
CLARKE, SE ;
AYRTON, AD ;
CHENERY, RJ .
XENOBIOTICA, 1994, 24 (06) :517-526
[3]   Microtiter plate assays for inhibition of human, drug-metabolizing cytochromes P450 [J].
Crespi, CL ;
Miller, VP ;
Penman, BW .
ANALYTICAL BIOCHEMISTRY, 1997, 248 (01) :188-190
[4]  
CRSPI CL, 1997, DRUG DRUG INTERACTIO, P171
[5]  
FDA,, 1997, GUID IND DISTEST I, P1
[6]   P450-ENZYMES - INHIBITION MECHANISMS, GENETIC-REGULATION AND EFFECTS OF LIVER-DISEASE [J].
MURRAY, M .
CLINICAL PHARMACOKINETICS, 1992, 23 (02) :132-146
[7]  
Obach RS, 1997, DRUG METAB DISPOS, V25, P1359
[8]   A POTENTIALLY HAZARDOUS INTERACTION BETWEEN ERYTHROMYCIN AND MIDAZOLAM [J].
OLKKOLA, KT ;
ARANKO, K ;
LUURILA, H ;
HILLER, A ;
SAARNIVAARA, L ;
HIMBERG, JJ ;
NEUVONEN, PJ .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1993, 53 (03) :298-305
[10]  
Rodrigues AD, 1997, DRUG METAB DISPOS, V25, P1097