共 50 条
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Discovery of N-(5,6-diarylpyridin-2-yl)amide derivatives as potent and selective A2B adenosine receptor antagonists
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Eastwood, Paul
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Gonzalez, Jacob
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Paredes, Sergio
;
Nueda, Arsenio
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Domenech, Teresa
;
Alberti, Joan
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Vidal, Bernat
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
2010, 20 (05)
:1697-1700

Eastwood, Paul
论文数: 0 引用数: 0
h-index: 0
机构:
Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain

Gonzalez, Jacob
论文数: 0 引用数: 0
h-index: 0
机构:
Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain

Paredes, Sergio
论文数: 0 引用数: 0
h-index: 0
机构:
Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain

Nueda, Arsenio
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h-index: 0
机构:
Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain

Domenech, Teresa
论文数: 0 引用数: 0
h-index: 0
机构:
Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain

Alberti, Joan
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h-index: 0
机构:
Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain

Vidal, Bernat
论文数: 0 引用数: 0
h-index: 0
机构:
Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain Almirall SA, Almirall Res Ctr, E-08980 Barcelona, Spain
[42]
Discovery and Optimization of a-Mangostin Derivatives as Novel PDE4 Inhibitors for the Treatment of Vascular Dementia
[J].
Liang, Jinhao
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Huang, Yi-You
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Zhou, Qian
;
Gao, Yuqi
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Li, Zhe
;
Wu, Deyan
;
Yu, Si
;
Guo, Lei
;
Chen, Zhen
;
Huang, Ling
;
Liang, Steven H.
;
He, Xixin
;
Wu, Ruibo
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Luo, Hai-Bin
.
JOURNAL OF MEDICINAL CHEMISTRY,
2020, 63 (06)
:3370-3380

Liang, Jinhao
论文数: 0 引用数: 0
h-index: 0
机构:
Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

Huang, Yi-You
论文数: 0 引用数: 0
h-index: 0
机构:
Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

Zhou, Qian
论文数: 0 引用数: 0
h-index: 0
机构:
Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

Gao, Yuqi
论文数: 0 引用数: 0
h-index: 0
机构:
Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

Li, Zhe
论文数: 0 引用数: 0
h-index: 0
机构:
Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

Wu, Deyan
论文数: 0 引用数: 0
h-index: 0
机构:
Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

Yu, Si
论文数: 0 引用数: 0
h-index: 0
机构:
Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

Guo, Lei
论文数: 0 引用数: 0
h-index: 0
机构:
Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

Chen, Zhen
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp, Dept Radiol, Div Nucl Med & Mol Imaging, Boston, MA 02114 USA
Harvard Med Sch, Boston, MA 02114 USA Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

Huang, Ling
论文数: 0 引用数: 0
h-index: 0
机构:
Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

Liang, Steven H.
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp, Dept Radiol, Div Nucl Med & Mol Imaging, Boston, MA 02114 USA
Harvard Med Sch, Boston, MA 02114 USA Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

He, Xixin
论文数: 0 引用数: 0
h-index: 0
机构:
Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

Wu, Ruibo
论文数: 0 引用数: 0
h-index: 0
机构:
Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China

Luo, Hai-Bin
论文数: 0 引用数: 0
h-index: 0
机构:
Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Guangzhou Univ Chinese Med, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China
[43]
Discovery and biological evaluation of N5-substituted 6,7-dioxo-6,7-dihydropteridine derivatives as potent Bruton's tyrosine kinase inhibitors
[J].
Chen, Haiyang
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Song, Peiran
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Diao, Yanyan
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Hao, Yongjia
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Dou, Dou
;
Wang, Wanqi
;
Fang, Xiaoyu
;
Wang, Yanling
;
Zhao, Zhenjiang
;
Ding, Jian
;
Li, Honglin
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Xie, Hua
;
Xu, Yufang
.
MEDCHEMCOMM,
2018, 9 (04)
:697-704

Chen, Haiyang
论文数: 0 引用数: 0
h-index: 0
机构:
East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China

Song, Peiran
论文数: 0 引用数: 0
h-index: 0
机构:
Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Div Antitumor Pharmacol, Shanghai 201203, Peoples R China
Univ Chinese Acad Sci, Beijing 100049, Peoples R China
ShanghaiTech Univ, Sch Life Sci & Technol, Shanghai 201210, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China

Diao, Yanyan
论文数: 0 引用数: 0
h-index: 0
机构:
East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China

Hao, Yongjia
论文数: 0 引用数: 0
h-index: 0
机构:
East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China

Dou, Dou
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h-index: 0
机构:
East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China

Wang, Wanqi
论文数: 0 引用数: 0
h-index: 0
机构:
East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China

Fang, Xiaoyu
论文数: 0 引用数: 0
h-index: 0
机构:
East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China

Wang, Yanling
论文数: 0 引用数: 0
h-index: 0
机构:
East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China

Zhao, Zhenjiang
论文数: 0 引用数: 0
h-index: 0
机构:
East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China

Ding, Jian
论文数: 0 引用数: 0
h-index: 0
机构:
Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Div Antitumor Pharmacol, Shanghai 201203, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China

Li, Honglin
论文数: 0 引用数: 0
h-index: 0
机构:
East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China

Xie, Hua
论文数: 0 引用数: 0
h-index: 0
机构:
Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Div Antitumor Pharmacol, Shanghai 201203, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China

Xu, Yufang
论文数: 0 引用数: 0
h-index: 0
机构:
East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioreactor Engn, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China
[44]
Discovery of furan and dihydrofuran-fused tricyclic benzo[d]imidazole derivatives as potent and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-1
[J].
Muthukaman, Nagarajan
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Tambe, Macchindra
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Deshmukh, Sanjay
;
Pisal, Dnyandeo
;
Tondlekar, Shital
;
Shaikh, Mahamadhanif
;
Sarode, Neelam
;
Kattige, Vidya G.
;
Pisat, Monali
;
Sawant, Pooja
;
Honnegowda, Srinivasa
;
Karande, Vikas
;
Kulkarni, Abhay
;
Behera, Dayanidhi
;
Jadhav, Satyawan B.
;
Sangana, Ramchandra R.
;
Gudi, Girish S.
;
Khairatkar-Joshi, Neelima
;
Gharat, Laxmikant A.
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
2017, 27 (23)
:5131-5138

Muthukaman, Nagarajan
论文数: 0 引用数: 0
h-index: 0
机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Tambe, Macchindra
论文数: 0 引用数: 0
h-index: 0
机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Deshmukh, Sanjay
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机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Pisal, Dnyandeo
论文数: 0 引用数: 0
h-index: 0
机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Tondlekar, Shital
论文数: 0 引用数: 0
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机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Shaikh, Mahamadhanif
论文数: 0 引用数: 0
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机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Sarode, Neelam
论文数: 0 引用数: 0
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机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Kattige, Vidya G.
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机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Biol Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Pisat, Monali
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h-index: 0
机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Biol Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Sawant, Pooja
论文数: 0 引用数: 0
h-index: 0
机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Biol Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Honnegowda, Srinivasa
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h-index: 0
机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Biol Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Karande, Vikas
论文数: 0 引用数: 0
h-index: 0
机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Biol Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Kulkarni, Abhay
论文数: 0 引用数: 0
h-index: 0
机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Biol Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Behera, Dayanidhi
论文数: 0 引用数: 0
h-index: 0
机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Drug Metab & Pharmacokinet, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Jadhav, Satyawan B.
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Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Drug Metab & Pharmacokinet, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Sangana, Ramchandra R.
论文数: 0 引用数: 0
h-index: 0
机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Drug Metab & Pharmacokinet, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Gudi, Girish S.
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h-index: 0
机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Drug Metab & Pharmacokinet, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Khairatkar-Joshi, Neelima
论文数: 0 引用数: 0
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机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Biol Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India

Gharat, Laxmikant A.
论文数: 0 引用数: 0
h-index: 0
机构:
Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India
[45]
Discovery of Novel 5-(Piperazine-1-carbonyl)pyridin-2(1H)-one Derivatives as Orally eIF4A3-Selective Inhibitors
[J].
Mizojiri, Ryo
;
Nakata, Daisuke
;
Satoh, Yoshihiko
;
Morishita, Daisuke
;
Shibata, Sachio
;
Iwatani-Yoshihara, Misa
;
Kosugi, Yohei
;
Kosaka, Mai
;
Takeda, Junpei
;
Sasaki, Shigekazu
;
Takami, Kazuaki
;
Fukuda, Koichiro
;
Kamaura, Masahiro
;
Sasaki, Shinobu
;
Arai, Ryosuke
;
Cary, Douglas R.
;
Imaeda, Yasuhiro
.
ACS MEDICINAL CHEMISTRY LETTERS,
2017, 8 (10)
:1077-1082

Mizojiri, Ryo
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Nakata, Daisuke
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan
Ono Pharmaceut Co Ltd, Osaka 6188585, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Satoh, Yoshihiko
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan
Astellas Pharma Inc, Tsukuba, Ibaraki 3058585, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Morishita, Daisuke
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Shibata, Sachio
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Iwatani-Yoshihara, Misa
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Kosugi, Yohei
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Kosaka, Mai
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Takeda, Junpei
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Sasaki, Shigekazu
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h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Takami, Kazuaki
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机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Fukuda, Koichiro
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan
Axcelead Drug Discovery Partners Inc, Fujisawa, Kanagawa 2518585, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Kamaura, Masahiro
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Sasaki, Shinobu
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan
Axcelead Drug Discovery Partners Inc, Fujisawa, Kanagawa 2518585, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Arai, Ryosuke
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan
Senjyu Pharmaceut Co Ltd, Osaka, Osaka 5410046, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Cary, Douglas R.
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan
PeptiDream Inc, Meguro Ku, Tokyo 1538904, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan

Imaeda, Yasuhiro
论文数: 0 引用数: 0
h-index: 0
机构:
Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan
[46]
Discovery of Novel Retigabine Derivatives as Potent KCNQ4 and KCNQ5 Channel Agonists with Improved Specificity
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Wang, Lei
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Qiao, Guan-Hua
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Hu, Hai-Ning
;
Gao, Zhao-Bing
;
Nan, Fa-Jun
.
ACS MEDICINAL CHEMISTRY LETTERS,
2019, 10 (01)
:27-33

Wang, Lei
论文数: 0 引用数: 0
h-index: 0
机构:
Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China
Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China

Qiao, Guan-Hua
论文数: 0 引用数: 0
h-index: 0
机构:
Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China
Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China

Hu, Hai-Ning
论文数: 0 引用数: 0
h-index: 0
机构:
Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China

Gao, Zhao-Bing
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h-index: 0
机构:
Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China

Nan, Fa-Jun
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h-index: 0
机构:
Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China
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Pharmacophore-Oriented Discovery of Novel 1,2,3-Benzotriazine-4-one Derivatives as Potent 4-Hydroxyphenylpyruvate Dioxygenase Inhibitors
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Yan, Yao-Chao
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Wu, Wei
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Huang, Guang-Yi
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Yang, Wen-Chao
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JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY,
2022, 70 (22)
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Yan, Yao-Chao
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h-index: 0
机构:
Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China

Wu, Wei
论文数: 0 引用数: 0
h-index: 0
机构:
Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China

Huang, Guang-Yi
论文数: 0 引用数: 0
h-index: 0
机构:
Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China

Yang, Wen-Chao
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h-index: 0
机构:
Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China

Chen, Qiong
论文数: 0 引用数: 0
h-index: 0
机构:
Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China

Qu, Ren-Yu
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h-index: 0
机构:
Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China

Lin, Hong-Yan
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h-index: 0
机构:
Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China

Yang, Guang-Fu
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h-index: 0
机构:
Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China Cent China Normal Univ, Int Joint Res Ctr Intelligent Biosensor Technol &, Key Lab Pesticide & Chem Biol, Minist Educ,Coll Chem, Wuhan 430079, Peoples R China
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Discovery of CZS-241: A Potent, Selective, and Orally Available Polo-Like Kinase 4 Inhibitor for the Treatment of Chronic Myeloid Leukemia
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Sun, Yin
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Liu, Hongbing
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Mu, Shuyi
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Sun, Pengkun
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Sun, Yu
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Wang, Lin
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Wang, Hanxun
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Wang, Jingkai
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Wu, Tianxiao
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Yin, Wenbo
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Qin, Qiaohua
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Sun, Yixiang
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JOURNAL OF MEDICINAL CHEMISTRY,
2023, 66 (04)
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Sun, Yin
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Xue, Yanli
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Liu, Hongbing
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharm, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Mu, Shuyi
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Sun, Pengkun
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Sun, Yu
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Wang, Lin
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Wang, Hanxun
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Wang, Jingkai
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Wu, Tianxiao
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Yin, Wenbo
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Qin, Qiaohua
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Sun, Yixiang
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Yang, Huali
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Zhao, Dongmei
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China

Cheng, Maosheng
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h-index: 0
机构:
Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Sch Pharmaceut Engn, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China
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Synthesis and biological evaluation of 5-carbamoyl-2-phenylpyrimidine derivatives as novel and potent PDE4 inhibitors
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Goto, Taiji
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Shiina, Akiko
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Mizukami, Kiyoshi
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2013, 21 (22)
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Goto, Taiji
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h-index: 0
机构:
Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan
Kyushu Univ, Grad Sch Pharmaceut Sci, Higashi Ku, Fukuoka 8128582, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan

Shiina, Akiko
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h-index: 0
机构:
Daiichi Sankyo Co Ltd, Qual & Safety Management Div, Chuo Ku, Tokyo 1038426, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan

Yoshino, Toshiharu
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h-index: 0
机构:
Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan

Mizukami, Kiyoshi
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h-index: 0
机构:
Daiichi Sankyo Co Ltd, Corp Strategy Div, Chuo Ku, Tokyo 1038426, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan

Hirahara, Kazuki
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h-index: 0
机构:
Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan

Suzuki, Osamu
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h-index: 0
机构:
Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan

Sogawa, Yoshitaka
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h-index: 0
机构:
Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan

Takahashi, Tomoko
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h-index: 0
机构:
Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan

Mikkaichi, Tsuyoshi
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h-index: 0
机构:
Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan

Nakao, Naoki
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h-index: 0
机构:
Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan

Takahashi, Mizuki
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h-index: 0
机构:
Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan

Hasegawa, Masashi
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h-index: 0
机构:
Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan

Sasaki, Shigeki
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h-index: 0
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Kyushu Univ, Grad Sch Pharmaceut Sci, Higashi Ku, Fukuoka 8128582, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan
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Design, synthesis, and biological evaluation of novel piperidine-4-carboxamide derivatives as potent CCR5 inhibitors
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EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,
2014, 71
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Hu, Suwen
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h-index: 0
机构:
Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China

Gu, Quan
论文数: 0 引用数: 0
h-index: 0
机构:
Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China

Wang, Zhilong
论文数: 0 引用数: 0
h-index: 0
机构:
Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China

Weng, Zhiyong
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h-index: 0
机构:
Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China

Cai, Yunrui
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h-index: 0
机构:
Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China

Dong, Xiaowu
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h-index: 0
机构:
Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China

Hu, Yongzhou
论文数: 0 引用数: 0
h-index: 0
机构:
Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China

Liu, Tao
论文数: 0 引用数: 0
h-index: 0
机构:
Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China

Xie, Xin
论文数: 0 引用数: 0
h-index: 0
机构:
Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China