An Efficient Synthesis of 5-Aryl-4,5-dihydro-3-(5-methyl-1-ptolyl-1H-1,2,3-triazol-4-yl)-1-(4-phenylthiazol-2-yl)pyrazoles

被引：4

作者：

Dong, Wang-Jun ^{[1
]}

Cui, Fu-Hong ^{[1
]}

Gao, Zhong-Lian ^{[1
]}

Li, Rong-Shan ^{[1
]}

Shen, Guo-Liang ^{[1
]}

Dong, Heng-Shan ^{[1
]}

机构：

[1] Lanzhou Univ, State Key Lab Appl Organ Chem, Inst Organ Chem, Coll Chem & Chem Engn, Lanzhou 730000, Gansu, Peoples R China

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2011年 / 48卷 / 05期

关键词：

SELECTIVE INHIBITORY-ACTIVITY; MONOAMINE-OXIDASE; PYRAZOLINE DERIVATIVES; AGENTS;

D O I：

10.1002/jhet.706

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Some new target products 5-aryl-4,5-dihydro-3-(5-methyl-1-p-tolyl-1H-1,2,3-triazol-4-yl)-1-(4-phenylthiazol-2-yl)pyrazoles 5a-j have been synthesized by reaction of 2-bromo-1-phenylethanone and compounds 4a-j which were prepared from the combination of thiosemicarbazide and (E)-3-aryl-1-(5methyl- 1-p-tolyl-1H-1,2,3-triazol-4-yl)-prop-2-en-1-ones 3a-j. All the structures were established by MS, IR, CHN, and H-1 NMR spectra data. Synthesis of structure diversity is applied.

引用

页码：1154 / 1160

页数：7

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