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- [41] The discovery of 2,5-isomers of triazole-pyrrolopyrimidine as selective Janus kinase 2 (JAK2) inhibitors versus JAK1 and JAK3BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 24 (21) : 5036 - 5046Lee, Sun-Mi论文数: 0 引用数: 0 h-index: 0机构: Gwangju Inst Sci & Technol GIST, Dept Med Syst Engn, 123 Cheomdan Gwagiro, Gwangju 61005, South Korea Gwangju Inst Sci & Technol GIST, Dept Med Syst Engn, 123 Cheomdan Gwagiro, Gwangju 61005, South KoreaYoon, Kyoung Bin论文数: 0 引用数: 0 h-index: 0机构: Gyeongsang Natl Univ, Coll Pharm, Jinju 52828, South Korea Gyeongsang Natl Univ, Pharmaceut Sci Res Inst, Jinju 52828, South Korea Gwangju Inst Sci & Technol GIST, Dept Med Syst Engn, 123 Cheomdan Gwagiro, Gwangju 61005, South KoreaLee, Hyo Jeong论文数: 0 引用数: 0 h-index: 0机构: Gyeongsang Natl Univ, Coll Pharm, Jinju 52828, South Korea Gyeongsang Natl Univ, Pharmaceut Sci Res Inst, Jinju 52828, South Korea Gwangju Inst Sci & Technol GIST, Dept Med Syst Engn, 123 Cheomdan Gwagiro, Gwangju 61005, South KoreaKim, Jiwon论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ, Coll Pharm, Seoul 08826, South Korea Seoul Natl Univ, Pharmaceut Sci Res Inst, Seoul 08826, South Korea Gwangju Inst Sci & Technol GIST, Dept Med Syst Engn, 123 Cheomdan Gwagiro, Gwangju 61005, South KoreaChung, You Kyoung论文数: 0 引用数: 0 h-index: 0机构: Ewha Womans Univ, Coll Pharm, Natl Leading Res Lab NLRL Mol Modeling & Drug Des, Seoul 03760, South Korea Ewha Womans Univ, Grad Sch Pharmaceut Sci, Seoul 03760, South Korea Gwangju Inst Sci & Technol GIST, Dept Med Syst Engn, 123 Cheomdan Gwagiro, Gwangju 61005, South KoreaCho, Won-Jea论文数: 0 引用数: 0 h-index: 0机构: Chonnam Natl Univ, Coll Pharm, Gwangju 61186, South Korea Chonnam Natl Univ, Res Inst Drug Dev, Gwangju 61186, South Korea Gwangju Inst Sci & Technol GIST, Dept Med Syst Engn, 123 Cheomdan Gwagiro, Gwangju 61005, South KoreaMukai, Chisato论文数: 0 引用数: 0 h-index: 0机构: Kanazawa Univ, Sch Pharm, Kakuma Machi, Kanazawa, Ishikawa 9201192, Japan Gwangju Inst Sci & Technol GIST, Dept Med Syst Engn, 123 Cheomdan Gwagiro, Gwangju 61005, South Korea论文数: 引用数: h-index:机构:Kang, Keon Wook论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ, Coll Pharm, Seoul 08826, South Korea Seoul Natl Univ, Pharmaceut Sci Res Inst, Seoul 08826, South Korea Gwangju Inst Sci & Technol GIST, Dept Med Syst Engn, 123 Cheomdan Gwagiro, Gwangju 61005, South Korea论文数: 引用数: h-index:机构:Ko, Hyojin论文数: 0 引用数: 0 h-index: 0机构: Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju, South Korea Gwangju Inst Sci & Technol GIST, Dept Med Syst Engn, 123 Cheomdan Gwagiro, Gwangju 61005, South KoreaKim, Yong-Chul论文数: 0 引用数: 0 h-index: 0机构: Gwangju Inst Sci & Technol GIST, Dept Med Syst Engn, 123 Cheomdan Gwagiro, Gwangju 61005, South Korea Gwangju Inst Sci & Technol GIST, Sch Life Sci, Gwangju, South Korea Gwangju Inst Sci & Technol GIST, Dept Med Syst Engn, 123 Cheomdan Gwagiro, Gwangju 61005, South Korea
- [42] ALTERNATING USE OF DIFFERENT JAK1/JAK2 INHIBITORS, A POSSIBLE THERAPEUTIC STRATEGY USEFUL IN PRIMARY MYELOFIBROSIS: A CASE REPORTHAEMATOLOGICA, 2020, 105 : 395 - 395Gutierrez, Lopez de Ocariz X.论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Hosp Univ 12 Octubre, Madrid, SpainVera, Guerrero E.论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Hosp Univ 12 Octubre, Madrid, SpainCarreno, Gomez-Tarragona G.论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Hosp Univ 12 Octubre, Madrid, SpainBuendia, Urena B.论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Hosp Univ 12 Octubre, Madrid, SpainDe Nicolas, Sol R.论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Hosp Univ 12 Octubre, Madrid, SpainHidalgo, Soto M.论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Hosp Univ 12 Octubre, Madrid, SpainLopez, Munoz N.论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Hosp Univ 12 Octubre, Madrid, SpainZamanillo, Herreros, I论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Hosp Univ 12 Octubre, Madrid, SpainIniguez, Garcia R.论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Hosp Univ 12 Octubre, Madrid, SpainPoza, Santaella M.论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Hosp Univ 12 Octubre, Madrid, SpainAyala, Diaz R.论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Hosp Univ 12 Octubre, Madrid, SpainMartinez, Lopez J.论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Hosp Univ 12 Octubre, Madrid, Spain
- [43] Role of JAK1, JAK2, and JAK3 in Functional Stimulation of Mesenchymal Precursor Cells by Alkaloid SongorineBulletin of Experimental Biology and Medicine, 2017, 163 : 443 - 446G. N. Zyuz’kov论文数: 0 引用数: 0 h-index: 0机构: E. D. Goldberg Research Institute of Pharmacology and Regenerative Medicine,Laboratory of Modeling of Physical Processes in Biology and MedicineE. V. Udut论文数: 0 引用数: 0 h-index: 0机构: E. D. Goldberg Research Institute of Pharmacology and Regenerative Medicine,Laboratory of Modeling of Physical Processes in Biology and MedicineL. A. Miroshnichenko论文数: 0 引用数: 0 h-index: 0机构: E. D. Goldberg Research Institute of Pharmacology and Regenerative Medicine,Laboratory of Modeling of Physical Processes in Biology and MedicineE. V. Simanina论文数: 0 引用数: 0 h-index: 0机构: E. D. Goldberg Research Institute of Pharmacology and Regenerative Medicine,Laboratory of Modeling of Physical Processes in Biology and MedicineT. Yu. Polyakova论文数: 0 引用数: 0 h-index: 0机构: E. D. Goldberg Research Institute of Pharmacology and Regenerative Medicine,Laboratory of Modeling of Physical Processes in Biology and MedicineL. A. Stavrova论文数: 0 引用数: 0 h-index: 0机构: E. D. Goldberg Research Institute of Pharmacology and Regenerative Medicine,Laboratory of Modeling of Physical Processes in Biology and MedicineV. V. Udut论文数: 0 引用数: 0 h-index: 0机构: E. D. Goldberg Research Institute of Pharmacology and Regenerative Medicine,Laboratory of Modeling of Physical Processes in Biology and MedicineM. Yu. Minakova论文数: 0 引用数: 0 h-index: 0机构: E. D. Goldberg Research Institute of Pharmacology and Regenerative Medicine,Laboratory of Modeling of Physical Processes in Biology and MedicineA. M. Dygai论文数: 0 引用数: 0 h-index: 0机构: E. D. Goldberg Research Institute of Pharmacology and Regenerative Medicine,Laboratory of Modeling of Physical Processes in Biology and MedicineA. V. Chaikovskii论文数: 0 引用数: 0 h-index: 0机构: E. D. Goldberg Research Institute of Pharmacology and Regenerative Medicine,Laboratory of Modeling of Physical Processes in Biology and MedicineV. I. Agafonov论文数: 0 引用数: 0 h-index: 0机构: E. D. Goldberg Research Institute of Pharmacology and Regenerative Medicine,Laboratory of Modeling of Physical Processes in Biology and MedicineV. V. Zhdanov论文数: 0 引用数: 0 h-index: 0机构: E. D. Goldberg Research Institute of Pharmacology and Regenerative Medicine,Laboratory of Modeling of Physical Processes in Biology and Medicine
- [44] 2,5-Isomers of triazole-pyrrolopyrimidine act as selective inhibitors of Janus kinase 2 (JAK2) compared to JAK1 and JAK3ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 252Sun-mi, Lee论文数: 0 引用数: 0 h-index: 0机构: GIST Gwang Ju Inst Sci & Technol, Dept Med Syst Engn, Gwang Ju, South Korea KRICT, Daejeon, South Korea GIST, Sch Life Sci, Gwangju, South KoreaKim, Yong-Chul论文数: 0 引用数: 0 h-index: 0机构: GIST, Sch Life Sci, Gwangju, South Korea GIST, Sch Life Sci, Gwangju, South Korea
- [45] The growth hormone receptor associates with Jak1, Jak2 and Tyk2 in human liverGROWTH HORMONE & IGF RESEARCH, 1999, 9 (03) : 212 - 218Hellgren, G论文数: 0 引用数: 0 h-index: 0机构: Gothenburg Univ, Sahlgrenska Univ Hosp, Dept Internal Med, Res Ctr Endocrinol & Metab, S-41345 Gothenburg, SwedenJansson, JO论文数: 0 引用数: 0 h-index: 0机构: Gothenburg Univ, Sahlgrenska Univ Hosp, Dept Internal Med, Res Ctr Endocrinol & Metab, S-41345 Gothenburg, SwedenCarlsson, LMS论文数: 0 引用数: 0 h-index: 0机构: Gothenburg Univ, Sahlgrenska Univ Hosp, Dept Internal Med, Res Ctr Endocrinol & Metab, S-41345 Gothenburg, SwedenCarlsson, B论文数: 0 引用数: 0 h-index: 0机构: Gothenburg Univ, Sahlgrenska Univ Hosp, Dept Internal Med, Res Ctr Endocrinol & Metab, S-41345 Gothenburg, Sweden Gothenburg Univ, Sahlgrenska Univ Hosp, Dept Internal Med, Res Ctr Endocrinol & Metab, S-41345 Gothenburg, Sweden
- [46] Preclinical characterization of atiprimod, a novel JAK2 AND JAK3 inhibitorInvestigational New Drugs, 2011, 29 : 818 - 826Alfonso Quintás-Cardama论文数: 0 引用数: 0 h-index: 0机构: UT MD Anderson Cancer Center,Department of LeukemiaTaghi Manshouri论文数: 0 引用数: 0 h-index: 0机构: UT MD Anderson Cancer Center,Department of LeukemiaZeev Estrov论文数: 0 引用数: 0 h-index: 0机构: UT MD Anderson Cancer Center,Department of LeukemiaDavid Harris论文数: 0 引用数: 0 h-index: 0机构: UT MD Anderson Cancer Center,Department of LeukemiaYing Zhang论文数: 0 引用数: 0 h-index: 0机构: UT MD Anderson Cancer Center,Department of LeukemiaAmos Gaikwad论文数: 0 引用数: 0 h-index: 0机构: UT MD Anderson Cancer Center,Department of LeukemiaHagop M. Kantarjian论文数: 0 引用数: 0 h-index: 0机构: UT MD Anderson Cancer Center,Department of LeukemiaSrdan Verstovsek论文数: 0 引用数: 0 h-index: 0机构: UT MD Anderson Cancer Center,Department of Leukemia
- [47] Discovery and Optimization of C-2 Methyl Imidazopyrrolopyridines as Potent and Orally Bioavailable JAK1 Inhibitors with Selectivity over JAK2JOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (13) : 6176 - 6193Zak, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAMendonca, Rohan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABalazs, Mercedesz论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABarrett, Kathy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABergeron, Philippe论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABlair, Wade S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAChang, Christine论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USADeshmukh, Gauri论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USADeVoss, Jason论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USADragovich, Peter S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAEigenbrot, Charles论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAGhilardi, Nico论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAGibbons, Paul论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAGradl, Stefan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHamman, Chris论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHanan, Emily J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHarstad, Eric论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Safety Assessment, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHewitt, Peter R.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHurley, Christopher A.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAJin, Tian论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, Shanghai 200131, Peoples R China Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAJohnson, Adam论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAJohnson, Tony论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAKenny, Jane R.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAKoehler, Michael F. T.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAKohli, Pawan Bir论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAKulagowski, Janusz J.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALabadie, Sharada论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALiao, Jiangpeng论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, Shanghai 200131, Peoples R China Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALiimatta, Marya论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALin, Zhonghua论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALupardus, Patrick J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAMaxey, Robert J.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAMurray, Jeremy M.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAPulk, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USARodriguez, Madeleine论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USASavage, Scott论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Small Mol Proc Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAShia, Steven论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USASteffek, Micah论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAUbhayakar, Savita论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAUltsch, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAvan Abbema, Anne论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAWard, Stuart I.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAXiao, Ling论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, Shanghai 200131, Peoples R China Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAXiao, Yisong论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, Shanghai 200131, Peoples R China Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA
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