Synthesis of 5-(3-hydroxypropyl)-7-methoxy-2-(3'-methoxy-4'-hydroxyphenyl)-3-benzo[b]furancarbaldehyde, a novel adenosine A(1) receptor ligand from the root of Salvia miltiorrhiza

被引：28

作者：

Kuo, YH ^{[1
]}

Wu, CH ^{[1
]}

机构：

[1] NATL RES INST CHINESE MED,TAIPEI,TAIWAN

来源：

JOURNAL OF NATURAL PRODUCTS | 1996年 / 59卷 / 06期

关键词：

D O I：

10.1021/np9603939

中图分类号：

Q94 [植物学];

学科分类号：

071001 ;

摘要：

A novel adenosine A(1) receptor ligand, 5-(3-hydroxypropyl)-7-methoxy-2-(3'-methoxy-4'-hydroxy- phenyl)-3-benzo[b]furancarbaldehyde (1), is a constituent of the roots of Salvia miltiorrhiza. Through biomimetic considerations, methyl ferulate was used as starting material for an eight-step synthesis of 1.

引用

页码：625 / 628

页数：4

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