Synthesis of N,N-disubstituted 3-amino-1,2,4-triazoles

被引：0
|
作者：
Katritzky, AR [1 ]
Rogovoy, BV
Vvedensky, VY
Kovalenko, K
Steel, PJ
Markov, VI
Forood, B
机构：
[1] Univ Florida, Dept Chem, Ctr Heterocycl Cpds, Gainesville, FL 32611 USA
[2] AE Arbuzov Organ & Phys Chem Inst, Kazan 420088, Russia
[3] Univ Canterbury, Dept Chem, Christchurch 1, New Zealand
[4] Ukrainian State Chem Technol Univ, UA-49005 Dniepropetrovsk, Ukraine
[5] Trega Biosci Inc, Exploratory Chem, San Diego, CA 92121 USA
来源：
SYNTHESIS-STUTTGART | 2001年 / 06期
关键词：
acylation; cyclization; regioselectivity; triazoles; benzotriazole; hydrazines;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A general method for the synthesis of N,N-disubstituted 3-amino-1,2,4-triazoles 5 from di(benzotriazolyl)methanimines 1 and 1', hydrazine and substituted hydrazines is developed. The desired compounds were prepared regioselectively under mild conditions by simple procedures in yields of up to 95%.
引用
收藏
页码：897 / 903
页数：7
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