Design of excitatory amino acid receptor agonists, partial agonists and antagonists: Ibotenic acid as a key lead structure

被引：54
作者：
KrogsgaardLarsen, P [1 ]
Ebert, B [1 ]
Lund, TM [1 ]
Brauner-Osborne, H [1 ]
Slok, FA [1 ]
Johansen, TN [1 ]
Brehm, L [1 ]
Madsen, U [1 ]
机构：
[1] ROYAL DANISH SCH PHARM, PHARMACOBIOTEC RES CTR, DEPT BIOL, DK-2100 COPENHAGEN, DENMARK
来源：
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 1996年 / 31卷 / 7-8期
关键词：
excitatory amino acid (EAA) receptor; ionotropic EAA receptor; metabotropic EAA receptor; AMPA agonist; AMPA partial agonist; AMPA antagonist; AMPA receptor modulator; kainic acid agonist; kainic acid antagonist; NMDA agonist; NMDA antagonist; glycine agonist; glycine partial agonist; glycine antagonist; metabotropic EAA agonist; metabotropic EAA antagonist; receptor autoradiography; functional partial agonism; EAA and neurodegeneration; EAA and schizophrenia; EAA and Alzheimer's disease;
D O I：
10.1016/0223-5234(96)89549-3
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
[No abstract available]
引用
收藏
页码：515 / 537
页数：23
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