Discovery and optimization of a novel series of thrombin receptor (PAR-1) antagonists: Potent, selective peptide mimetics based on indole and indazole templates

被引：75
作者：
Zhang, HC [1 ]
Derian, CK
Andrade-Gordon, P
Hoekstra, WJ
McComsey, DF
White, KB
Poulter, BL
Addo, MF
Cheung, WM
Damiano, BP
Oksenberg, D
Reynolds, EE
Pandey, A
Scarborough, RM
Maryanoff, BE
机构：
[1] RW Johnson Pharmaceut Res Inst, Spring House, PA 19477 USA
[2] COR Therapeut Inc, S San Francisco, CA 94080 USA
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 2001年 / 44卷 / 07期
关键词：
D O I：
10.1021/jm000506s
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：1021 / 1024
页数：4
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