Synthesis of C3-Modified Carbapenems

被引:0
作者
Torosyan, S. A. [1 ]
Nuriakhmetova, Z. F. [1 ]
Gimalova, F. A. [1 ]
Miftakhov, M. S. [1 ]
机构
[1] Russian Acad Sci, Ufa Inst Chem, Ufa Fed Res Ctr, Ufa 450054, Russia
基金
俄罗斯科学基金会;
关键词
2-ethoxy-1; 3-oxathiolan-5-one; thiols; carbapenem enol phosphate; substitution reactions; carbapenems;
D O I
10.1134/S1070428020010029
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Reactions of 4-nitrobenzyl (4R,5R,6S)-3-[(diphenoxyphosphoryl)oxy]-6-[(1R)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylate with 2-sulfanylacetamides derived from taurine and cytisine afforded the corresponding products of Ad(N)E substitution of the diphenoxyphosphoryl group.
引用
收藏
页码:7 / 10
页数:4
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