Synthesis of C3-Modified Carbapenems

被引：0
作者：
Torosyan, S. A. [1 ]
Nuriakhmetova, Z. F. [1 ]
Gimalova, F. A. [1 ]
Miftakhov, M. S. [1 ]
机构：
[1] Russian Acad Sci, Ufa Inst Chem, Ufa Fed Res Ctr, Ufa 450054, Russia
来源：
RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2020年 / 56卷 / 01期
基金：
俄罗斯科学基金会;
关键词：
2-ethoxy-1; 3-oxathiolan-5-one; thiols; carbapenem enol phosphate; substitution reactions; carbapenems;
D O I：
10.1134/S1070428020010029
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Reactions of 4-nitrobenzyl (4R,5R,6S)-3-[(diphenoxyphosphoryl)oxy]-6-[(1R)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylate with 2-sulfanylacetamides derived from taurine and cytisine afforded the corresponding products of Ad(N)E substitution of the diphenoxyphosphoryl group.
引用
收藏
页码：7 / 10
页数：4
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