Solid phase synthesis of 1,2-disubstituted alkenes: A novel alkynyldihydropyridine to alkenylpyridine isomerization

被引：5

作者：

Chen, CX ^{[1
]}

Wang, BW ^{[1
]}

Munoz, B ^{[1
]}

机构：

[1] Merck Res Labs, San Diego, CA 92131 USA

来源：

SYNLETT | 2003年 / 15期

关键词：

solid-phase synthesis; 1,2-disubstituted alkenes; alkynyldihydropyridine; alkenylpyridine; isomerization;

D O I：

10.1055/s-2003-43343

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A series of 1,2-disubstituted pyridylalkenes have been prepared using a solid-phase resin approach. This approach takes advantage of a novel alkynyldihydropyridine to alkenylpyridine isomerization.

引用

页码：2404 / 2406

页数：3

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