Synthesis of novel thiazolo[5,4-d]pyrimidines

被引：0

作者：

Chattopadhyay, Gautam ^{[1
]}

Saha, Debnath ^{[1
]}

Ray, Partha Sinha ^{[1
]}

Naskar, Subhendu ^{[1
]}

Sarkar, Swarbhanu ^{[1
]}

机构：

[1] Presidency Coll, Postgrad Dept Chem, Kolkata 700073, India

来源：

INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 2010年 / 49卷 / 09期

关键词：

Thiazolo[5,4-d]pyrimidines; mesoionic isomer; heteroaryl motif's; aminothiazolecarboxamide;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

2-Methylsulphany1-5-aminothiazole-4-carboxamide 1 has been used as a convenient precursor for the synthesis of new thiazolo[4.5-e][1,2,4-triazoloirl][4,3-c]pyrimidines 5 and the corresponding tetrazolo analogue 7. A mesoionic isomer 8 seems to exist along with 7. Interesting heteroarylthiazolo pyrimidirte motifs have also been prepared via suitably substituted thiazolo[5.4-d]pyrimidines.

引用

页码：1229 / 1234

页数：6

共 50 条

[21] Regioselective synthesis of substituted isoxozolo[5,4-d]pyrimidines
Alyabiev, Sergey B.
Kravchenko, Dmitri V.
Ivachtchenko, Alexandre V.
MENDELEEV COMMUNICATIONS, 2008, 18 (03) : 144 - 146
[22] STUDIES ON CONDENSED PYRIMIDINE SYSTEMS .4. SOME THIAZOLO[5,4-D]PYRIMIDINES
FALCO, EA
HITCHINGS, GH
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1950, 72 (07) : 3203 - 3205
[23] REACTION OF BISCYANINE CHROMOPHORES FROM THIAZOLO-[5,4-D] [5,4-D] THIAZOLE
MIKHAILENKO, FA
ISHCHENKO, II
UKRAINSKII KHIMICHESKII ZHURNAL, 1974, 40 (12): : 1331 - 1333
[24] Design and Synthesis of Novel Thiazolo[5,4-d]pyrimidine Derivatives as Potential Angiogenesis Inhibitors
Xue, Wen-Jun
Du, Jian-Yao
Deng, Ya-Hui
Yan, Zhong-Hui
Liu, Ji-Ping
Liu, Yu
Sun, Li-Ping
CHEMISTRY & BIODIVERSITY, 2019, 16 (08)
[25] SYNTHESIS OF BICYCLIC NUCLEOSIDES RELATED TO URIDINE, 4-(BETA-D-RIBOFURANOSYL)THIAZOLO[5,4-D]PYRIMIDINES
SCHMIDT, CL
RUSHO, WJ
TOWNSEND, LB
JOURNAL OF THE CHEMICAL SOCIETY D-CHEMICAL COMMUNICATIONS, 1971, (23): : 1515 - &
[26] ISOTHIAZOLES .3. SYNTHESIS OF ISOTHIAZOLO[5,4-D]PYRIMIDINES
ANDERSON, RC
HSIAO, YY
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1975, 12 (05) : 883 - 887
[27] UBER EINIGE THIAZOLO[5,4-D]PYRIMIDINE
VONHAHN, H
PRIJS, B
ERLENMEYER, H
HELVETICA CHIMICA ACTA, 1956, 39 (02) : 341 - 347
[28] SYNTHESIS AND PROPERTIES OF THIAZOLO[5,4-D]PYRIMIDINE 1-OXIDES
SENGA, K
ICHIBA, M
KANAZAWA, H
NISHIGAKI, S
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1982, 19 (01) : 77 - 80
[29] Synthesis of pyrrolino[3,4-d]pyrazoles, pyrazoles, pyrazolo[5,4-d]pyrimidines and pyrazolo[3,4-d]pyrimidines
Riheem, Nadia A. Abdel
Rateb, Nora M.
Eldin, Sanaa M.
DRUGS OF THE FUTURE, 2007, 32 : 40 - 41
[30] A one step synthesis of 1-alkylpyrazolo[5,4-d]pyrimidines
Boyd, Scott
Campbell, Leonie
Liao, Wensheng
Meng, Qinghong
Peng, Zuozhong
Wan, Xiaoping
Waring, Michael J.
TETRAHEDRON LETTERS, 2008, 49 (52) : 7395 - 7397

← 1 2 3 4 5 →