Synthesis, structure and bioactivity of nitrobenzoimidazole derivatives

被引：0

作者：

Wang, LY ^{[1
]}

Gao, Y ^{[1
]}

Yang, BQ ^{[1
]}

Zhen, S ^{[1
]}

机构：

[1] NW Univ Xian, Dept Chem, Xian 710069, Peoples R China

来源：

CHEMICAL JOURNAL OF CHINESE UNIVERSITIES-CHINESE | 2005年 / 26卷 / 12期

关键词：

nitrobenzoimidazole; synthesis; crystal structure; antimicrobial activity;

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

It was reported that benzoimidazole and ferrocene compounds maybe exhibit high pharmaceutical functions. Eight new nitrobenzoimidazole derivatives were prepared by the reaction of ferrocene sulfonylchloride with 5-nitrobenzoimidazole and characterized by means of elemental analysis, MS and H-1 NMR. The structure of the new compounds was further confirmed by X-ray crystallograghic analysis as exemplified by compounds 3b. The activities of compounds 3a-4d were evaluated against five fungicides. Compared with carbendazim(50% wet powder), better inhibitory activities were observed for these synthesized compounds.

引用

页码：2241 / 2246

页数：6

共 14 条

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