Strategies for the Design of HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: Lessons from the Development of Seven Representative Paradigms

被引：118
作者：
Li, Dongyue [1 ]
Zhan, Peng [1 ]
De Clercq, Erik [2 ]
Liu, Xinyong [1 ]
机构：
[1] Shandong Univ, Sch Pharmaceut Sci, Dept Med Chem, Jinan 250012, Shandong, Peoples R China
[2] Katholieke Univ Leuven, Rega Inst Med Res, B-3000 Louvain, Belgium
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 2012年 / 55卷 / 08期
基金：
中国国家自然科学基金; 中国博士后科学基金; 高等学校博士学科点专项科研基金;
关键词：
RESISTANT MUTANT VIRUSES; MEDICINAL CHEMISTRY; DRUG CANDIDATES; MOLECULAR HYBRIDIZATION; ANGSTROM RESOLUTION; ANTIVIRAL ACTIVITY; ETRAVIRINE TMC125; BROAD POTENCY; DAPY ANALOGS; WILD-TYPE;
D O I：
10.1021/jm200990c
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
[No abstract available]
引用
收藏
页码：3595 / 3613
页数：19
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