Lutetium-177 Therapeutic Radiopharmaceuticals: Linking Chemistry, Radiochemistry, and Practical Applications

被引:245
作者
Banerjee, Sharmila [1 ]
Pillai, M. R. A. [2 ]
Knapp, F. F. [3 ]
机构
[1] BARC, Radiopharmaceut Chem Sect, Bombay 400085, Maharashtra, India
[2] Mol Grp Co, Ernakulam 682508, Kerala, India
[3] Oak Ridge Natl Lab, Med Radioisotope Program, Oak Ridge, TN 37830 USA
关键词
STIMULATING HORMONE PEPTIDE; IN-VIVO EVALUATION; PRELIMINARY BIOLOGICAL EVALUATION; RADIOLABELED SOMATOSTATIN ANALOG; RECEPTOR RADIONUCLIDE THERAPY; CARRIER-ADDED LU-177; LU-177-LABELED GOLD NANOPARTICLES; LONG-TERM TOXICITY; GRP-R AGONIST; MONOCLONAL-ANTIBODY;
D O I
10.1021/cr500171e
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
[No abstract available]
引用
收藏
页码:2934 / 2974
页数:41
相关论文
共 294 条
[1]   Preliminary studies on 177Lu-labeled sodium pyrophosphate (177Lu-PYP) as a potential bone-seeking radiopharmaceutical for bone pain palliation [J].
Abbasi, Imtiaz Ahmed .
NUCLEAR MEDICINE AND BIOLOGY, 2012, 39 (06) :763-769
[2]   Studies on 177Lu-labeled methylene diphosphonate as potential bone-seeking radiopharmaceutical for bone pain palliation [J].
Abbasi, Imtiaz Ahmed .
NUCLEAR MEDICINE AND BIOLOGY, 2011, 38 (03) :417-425
[3]   177Lu-EDTMP for palliation of pain from bone metastases in patients with prostate and breast cancer: a phase II study [J].
Agarwal, Krishan Kant ;
Singla, Suhas ;
Arora, Geetanjali ;
Bal, Chandrasekhar .
EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2015, 42 (01) :79-88
[4]   In vitro and in vivo characterization of 177Lu-huA33 A radioimmunoconjugate against colorectal cancer [J].
Almqvist, Ylva ;
Steffen, Ann-Charlott ;
Tolmachev, Vladimir ;
Divgi, Chaitanya R. ;
Sundin, Anders .
NUCLEAR MEDICINE AND BIOLOGY, 2006, 33 (08) :991-998
[5]   Intraperitoneal radioimmunotherapy of ovarian cancer with Lu-177-CC49: A phase I/II study [J].
Alvarez, RD ;
Partridge, EE ;
Khazaeli, MB ;
Plott, G ;
Austin, M ;
Kilgore, L ;
Russell, CD ;
Liu, TP ;
Grizzle, WE ;
Schlom, J ;
LoBuglio, AF ;
Meredith, RF .
GYNECOLOGIC ONCOLOGY, 1997, 65 (01) :94-101
[6]   Radiopeptide Imaging and Therapy in Europe [J].
Ambrosini, Valentina ;
Fani, Melpomeni ;
Fanti, Stefano ;
Forrer, Flavio ;
Maecke, Helmut R. .
JOURNAL OF NUCLEAR MEDICINE, 2011, 52 :42S-55S
[7]   ISOLATION AND STRUCTURE OF BOMBESIN AND ALYTESIN, 2 ANALOGOUS ACTIVE PEPTIDES FROM SKIN OF EUROPEAN AMPHIBIANS BOMBINA AND ALYTES [J].
ANASTASI, A ;
ERSPAMER, V ;
BUCCI, M .
EXPERIENTIA, 1971, 27 (02) :166-&
[8]   THE TREATMENT OF MYELOMATOSIS WITH LUTECIUM-177 [J].
ANDERSON, J ;
FARMER, FT ;
HAGGITH, JW ;
HILL, M .
BRITISH JOURNAL OF RADIOLOGY, 1960, 33 (390) :374-378
[9]   177Lu-EDTMP:: A potential therapeutic bone agent [J].
Ando, A ;
Ando, I ;
Tonami, N ;
Kinuya, S ;
Kazuma, K ;
Kataiwa, A ;
Nakagawa, M ;
Fujita, N .
NUCLEAR MEDICINE COMMUNICATIONS, 1998, 19 (06) :587-591
[10]   Outcome of treating advanced neuroendocrine tumours with radiolabelled somatostatin analogues [J].
Angustias Muros, Maria ;
Varsavsky, Mariela ;
Iglesias Rozas, Pablo ;
Valdivia, Javier ;
Ramon Delgado, Juan ;
Forrer, Flavio ;
Bodei, Lisa ;
Paganelli, Giovanni .
CLINICAL & TRANSLATIONAL ONCOLOGY, 2009, 11 (01) :48-53