SYNTHESIS OF SOME NOVEL FUSED AZOLE DERIVATIVES

被引：21
|
作者：
Soliman, A. M. [1 ]
Sultan, A. A. [1 ]
El Remaily, M. A. A. [1 ]
Abdel-Ghany, H. [1 ]
机构：
[1] Sohag Univ, Fac Sci, Dept Chem, Sohag, Egypt
来源：
SYNTHETIC COMMUNICATIONS | 2012年 / 42卷 / 18期
关键词：
Isocyanate; phenylisothiocyanate; pyrazolopyridine; pyrazolopyrimidine; ANTIMICROBIAL ACTIVITY; HETEROCYCLES;
D O I：
10.1080/00397911.2011.566462
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A novel synthesis of pyrazolopyrimidine derivatives was reported wherein 5-amino-1-benzoyl-3-(methylthio)-1H-pyrazole-4-carbonitrile was treated with formic acid, formamide, thioacetamide, carbon disulfide, and phenylisocyanate and phenylisothiocyanate.
引用
收藏
页码：2748 / 2762
页数：15
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