Identification of enantiomerically pure 5-HT6 receptor antagonists by chiral resolution

被引：0
|
作者：
Park, Chul Min [1 ]
Kang, Sunhee [1 ]
Park, Wookyu [2 ]
Park, Nosang [1 ]
Seong, Churlmin [1 ]
机构：
[1] Korea Res Inst Chem Technol, Div Bioorgan, CNS Res Team, Taejon 305606, South Korea
[2] Korea Res Inst Chem Technol, Pharmaceut Screening Res Team, Taejon 305606, South Korea
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2007年 / 233卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
294-MEDI
引用
收藏
页码：697 / 697
页数：1
相关论文
共 50 条
  • [1] Potent and selective 5-HT6 receptor antagonists
    Bromidge, SM
    MEDICINAL CHEMISTRY INTO THE MILLENNIUM, 2001, (264): : 101 - 119
  • [2] IDENTIFICATION OF NOVEL INDANYLAMIDINOHYDRAZONES AS 5-HT6 ANTAGONISTS
    Mesquida, Neus
    Lopez-Perez, Sara
    Dinares, Immaculada
    Frigola, Jordi
    Merce, Ramon
    Holenz, Joerg
    Perez, Raquel
    Burgueno, Javier
    Alcalde, Ermitas
    DRUGS OF THE FUTURE, 2009, 34 : 126 - 126
  • [3] Identification of Novel Indanylsulfonamide Guanylhydrazones as Potent 5-HT6 Serotonin Receptor Antagonists
    Mesquida, Neus
    Lopez-Perez, Sara
    Dinares, Immaculada
    Frigola, Jordi
    Merce, Ramon
    Holenz, Joerg
    Perez, Raquel
    Burgueno, Javier
    Alcalde, Ermitas
    JOURNAL OF MEDICINAL CHEMISTRY, 2009, 52 (19) : 6153 - 6157
  • [4] Cognitive enhancing properties of 5-HT6 receptor antagonists
    Chuang, TT
    Rogers, DC
    Hagan, JJ
    Lacroix, LP
    Dawson, LA
    Foley, AG
    Regan, CM
    Heidbreder, CA
    Upton, N
    INTERNATIONAL JOURNAL OF NEUROPSYCHOPHARMACOLOGY, 2004, 7 : S14 - S14
  • [5] Potent and selective 5-HT6 receptor antagonists.
    Bromidge, SM
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1999, 218 : U971 - U971
  • [6] Novel 5-HT6 receptor antagonists for the treatment of obesity
    Shacham, S
    Marantz, Y
    Senderowitz, H
    Orbach, P
    Sharadendu, A
    Becker, O
    Noiman, S
    OBESITY RESEARCH, 2005, 13 : A192 - A192
  • [7] 5-HT6 Receptor Antagonists as Potential Therapeutics for Cognitive Impairment
    Rosse, Gerard
    Schaffhauser, Herve
    CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2010, 10 (02) : 207 - 221
  • [8] Novel brain penetrant benzofuropiperidine 5-HT6 receptor antagonists
    Sundar, Babu G.
    Bailey, Thomas R.
    Dunn, Derek D.
    Bacon, Edward R.
    Salvino, Joseph M.
    Morton, George C.
    Aimone, Lisa D.
    Huang Zeqi
    Mathiasen, Joanne R.
    Dicamillo, Amy
    Huffman, Mark J.
    McKenna, Beth A.
    Kopec, Karla
    Lu, Lily D.
    Brown, Rebecca
    Qian, Jie
    Angeles, Thelma
    Connors, Thomas
    Spais, Chrysanthe
    Holskin, Beverly
    Galinis, Deborah
    Duzic, Emir
    Schaffhauser, Herve
    Rosse, Gerard C.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (01) : 120 - 123
  • [9] Bicyclic piperazinylbenzenesulphonamides are potent and selective 5-HT6 receptor antagonists
    Bromidge, SM
    Clarke, SE
    King, FD
    Lovell, PJ
    Newman, H
    Riley, G
    Routledge, C
    Serafinowska, HT
    Smith, DR
    Thomas, DR
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2002, 12 (10) : 1357 - 1360
  • [10] 5-HT6 receptor antagonist
    Lloyd, AW
    DRUG DISCOVERY TODAY, 1999, 4 (05) : 238 - 238
12345