Palladium-catalyzed intermolecular α-arylation of N-protected 2-piperidinones

被引：59
|
作者：
Cossy, J [1 ]
de Filippis, A [1 ]
Pardo, DG [1 ]
机构：
[1] Ecole Super Phys & Chim Ind Ville Paris, CNRS, Chim Organ Lab, F-75231 Paris 05, France
来源：
ORGANIC LETTERS | 2003年 / 5卷 / 17期
关键词：
D O I：
10.1021/ol0350036
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
graphic The alpha-arylation of the zinc enolate of N-protected 2-piperidinones with aryl bromides in the presence of a palladium catalyst is described as a general method.
引用
收藏
页码：3037 / 3039
页数：3
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