A new approach to the synthesis of benzo[b][1,8]naphthyridin-4(1H)ones.

被引:0
|
作者
Vijayalakshmi, S [1 ]
Ragunath, L [1 ]
Rajendran, SP [1 ]
机构
[1] Bharathiar Univ, Dept Chem, Coimbatore 641046, Tamil Nadu, India
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中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Condensation of 3-acetyl-4-phenylquinoline-2(1H)ones I with benzalclehydes give 4-phenyl-3cinnamoylquinolin-2(1H)ones 2 which inturn were converted to 2-chloro-3-cinnamoyl-4-phenylquinolines. 3. Compounds 3 were then aminated with p-aminobenzensulfonamide and then subjected to bromination-dehydrobromination step to yield 2,5-diphenylbenzo[b][1,8]naphthyridin-4(1H)ones 5.
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页码:177 / 182
页数:6
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