Cytochrome P450 3A pharmacogenetics: the road that needs traveled

被引:35
作者
Flockhart, DA
Rae, JM
机构
[1] Indiana Univ, Sch Med, Div Clin Pharmacol, Indianapolis, IN USA
[2] Univ Michigan, Med Ctr, Div Hematol & Oncol, Ann Arbor, MI USA
关键词
D O I
10.1038/sj.tpj.6500144
中图分类号
Q3 [遗传学];
学科分类号
071007 ; 090102 ;
摘要
[No abstract available]
引用
收藏
页码:3 / 5
页数:3
相关论文
共 26 条
[1]   POLYMORPHIC HYDROXYLATION OF S-MEPHENYTOIN AND OMEPRAZOLE METABOLISM IN CAUCASIAN AND CHINESE SUBJECTS [J].
ANDERSSON, T ;
REGARDH, CG ;
LOU, YC ;
ZHANG, Y ;
DAHL, ML ;
BERTILSSON, L .
PHARMACOGENETICS, 1992, 2 (01) :25-31
[2]   Population distribution and effects on drug metabolism of a genetic variant in the 5′ promotor region of CYP3A4 [J].
Ball, SE ;
Scatina, JA ;
Kao, J ;
Ferron, GM ;
Fruncillo, R ;
Mayer, P ;
Weinryb, I ;
Guida, M ;
Hopkins, PJ ;
Warner, N ;
Hall, J .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1999, 66 (03) :288-294
[3]   INHIBITION BY PAROXETINE OF DESIPRAMINE METABOLISM IN EXTENSIVE BUT NOT IN POOR METABOLIZERS OF SPARTEINE [J].
BROSEN, K ;
HANSEN, JG ;
NIELSEN, KK ;
SINDRUP, SH ;
GRAM, LF .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1993, 44 (04) :349-355
[4]   Molecular mechanisms of polymorphic CYP3A7 expression in adult human liver and intestine [J].
Burk, O ;
Tegude, H ;
Koch, I ;
Hustert, E ;
Wolbold, R ;
Glaeser, H ;
Klein, K ;
Fromm, MF ;
Nuessler, AK ;
Neuhaus, P ;
Zanger, UM ;
Eichelbaum, M ;
Wojnowski, L .
JOURNAL OF BIOLOGICAL CHEMISTRY, 2002, 277 (27) :24280-24288
[5]  
Caraco Y, 1999, J PHARMACOL EXP THER, V290, P413
[6]   10-hydroxylation of nortriptyline in white persons with 0, 1, 2, 3, and 13 functional CΥP2D6 genes [J].
Dalén, P ;
Dahl, ML ;
Ruiz, MLB ;
Nordin, J ;
Bertilsson, L .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1998, 63 (04) :444-452
[7]   Identification and functional characterization of eight CYP3A4 protein variants [J].
Eiselt, R ;
Domanski, TL ;
Zibat, A ;
Mueller, R ;
Presecan-Siedel, E ;
Hustert, E ;
Zanger, UM ;
Brockmoller, J ;
Klenk, HP ;
Meyer, UA ;
Khan, KK ;
He, YA ;
Halpert, JR ;
Wojnowski, L .
PHARMACOGENETICS, 2001, 11 (05) :447-458
[8]   Association of CYP3A4 genotype with treatment-related leukemia [J].
Felix, CA ;
Walker, AH ;
Lange, BJ ;
Williams, TM ;
Winick, NJ ;
Cheung, NKV ;
Lovett, BD ;
Nowell, PC ;
Blair, IA ;
Rebbeck, TR .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1998, 95 (22) :13176-13181
[9]   The human cytochrome P450 3A locus. Gene evolution by capture of downstream exons [J].
Finta, C ;
Zaphiropoulos, PG .
GENE, 2000, 260 (1-2) :13-23
[10]   Effect of genetic differences in omeprazole metabolism on cure rates for Helicobacter pylori infection and peptic ulcer [J].
Furuta, T ;
Ohashi, K ;
Kamata, T ;
Takashima, M ;
Kosuge, K ;
Kawasaki, T ;
Hanai, H ;
Kubota, T ;
Ishizaki, T ;
Kaneko, E .
ANNALS OF INTERNAL MEDICINE, 1998, 129 (12) :1027-1030