A Facile Synthesis of 1-(4-Methoxybenzyl)-4-[(E)-4-(trimethylsilyl)but-1-en-3-yn-1-yl]-1H-indole and 2-Aryl-1-(4-methoxybenzyl)-1H-indole-4-carbaldehydes

被引:0
作者
Karuna, Ch. [1 ]
Reddy, Ch. V. R. [1 ]
Laxminarayana, E. [2 ]
机构
[1] Jawaharlal Nehru Technol Univ Hyderabad, Dept Chem, Hyderabad 500085, India
[2] Sreenidhi Inst Sci & Technol Autonomous Yamnampet, Dept Chem, Hyderabad 501301, India
关键词
4-bromoindole; enyne group; 3-formylindoles; TBDMS-Cl; indole-4-carbaldehydes; INDOLE-DERIVATIVES; BIOLOGICAL EVALUATION; DESIGN; PHARMACOPHORE; ANTIOXIDANT; AGENTS;
D O I
10.1134/S1070428022100190
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Indole derivatives containing a enyne moiety are precursors to many indole-based natural products like indiacen. These scaffolds were synthesized from commercially available 4-bromoindole and other inex-pensive reagents. The synthesized compounds were characterized by spectral data.
引用
收藏
页码:1516 / 1519
页数:4
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