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Bone-targeted, nonpeptide inhibitors of the Src SH2 domain: Structure-based design and structure-activity relationships
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Bohacek, R
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0
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0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Bohacek, R
[
1
]
Weigele, M
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0
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0
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0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Weigele, M
[
1
]
Jacobsen, V
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0
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0
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0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Jacobsen, V
[
1
]
Macek, K
论文数:
0
引用数:
0
h-index:
0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Macek, K
[
1
]
Luke, G
论文数:
0
引用数:
0
h-index:
0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Luke, G
[
1
]
Sundaramoorthi, R
论文数:
0
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0
h-index:
0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Sundaramoorthi, R
[
1
]
Metcalf, C
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0
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0
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0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Metcalf, C
[
1
]
Shakespeare, W
论文数:
0
引用数:
0
h-index:
0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Shakespeare, W
[
1
]
Yang, M
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Yang, M
[
1
]
Wang, YH
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Wang, YH
[
1
]
Kawahata, N
论文数:
0
引用数:
0
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0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Kawahata, N
[
1
]
Takeuchi, C
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0
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0
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0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Takeuchi, C
[
1
]
Haraldson, C
论文数:
0
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0
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0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Haraldson, C
[
1
]
Varkhedkar, V
论文数:
0
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0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Varkhedkar, V
[
1
]
Johnson, D
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0
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0
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0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Johnson, D
[
1
]
Hatada, M
论文数:
0
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0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Hatada, M
[
1
]
Lu, XD
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Lu, XD
[
1
]
Narula, S
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Narula, S
[
1
]
Eyermann, C
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Eyermann, C
[
1
]
Violette, S
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Violette, S
[
1
]
Bartlett, C
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Bartlett, C
[
1
]
Guan, W
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Guan, W
[
1
]
Smith, J
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Smith, J
[
1
]
Adams, S
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Adams, S
[
1
]
Lynch, B
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Lynch, B
[
1
]
MacNeil, I
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
MacNeil, I
[
1
]
van Schravendijk, MR
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
van Schravendijk, MR
[
1
]
Stebbins, K
论文数:
0
引用数:
0
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0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Stebbins, K
[
1
]
Wood, S
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0
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0
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0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Wood, S
[
1
]
Li, P
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Li, P
[
1
]
Yuan, R
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Yuan, R
[
1
]
Dalgarno, D
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Dalgarno, D
[
1
]
Cerasoli, F
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Cerasoli, F
[
1
]
Sawyer, T
论文数:
0
引用数:
0
h-index:
0
机构:
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Sawyer, T
[
1
]
机构
:
[1]
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
来源
:
PEPTIDES FOR THE NEW MILLENNIUM
|
2000年
关键词
:
D O I
:
暂无
中图分类号
:
Q5 [生物化学];
Q7 [分子生物学];
学科分类号
:
071010 ;
081704 ;
摘要
:
引用
收藏
页码:558 / 560
页数:3
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[5]
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WARNER LAMBERT PARKE DAVIS, PARKE DAVIS PHARMACEUT RES DIV, DEPT BIOCHEM, ANN ARBOR, MI 48105 USA
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0
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WARNER LAMBERT PARKE DAVIS, PARKE DAVIS PHARMACEUT RES DIV, DEPT BIOCHEM, ANN ARBOR, MI 48105 USA
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WARNER LAMBERT PARKE DAVIS, PARKE DAVIS PHARMACEUT RES DIV, DEPT BIOCHEM, ANN ARBOR, MI 48105 USA
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0
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WARNER LAMBERT PARKE DAVIS, PARKE DAVIS PHARMACEUT RES DIV, DEPT BIOCHEM, ANN ARBOR, MI 48105 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Buchanan, JL
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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Structure-based design of a novel series of nonpeptide ligands that bind to the pp60src SH2 domain
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Parke Davis Pharmaceut Res, Dept Chem, Ann Arbor, MI 48106 USA
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Parke Davis Pharmaceut Res, Dept Chem, Ann Arbor, MI 48106 USA
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Parke Davis Pharmaceut Res, Dept Chem, Ann Arbor, MI 48106 USA
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Parke Davis Pharmaceut Res, Dept Chem, Ann Arbor, MI 48106 USA
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Parke Davis Pharmaceut Res, Dept Chem, Ann Arbor, MI 48106 USA
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Parke Davis Pharmaceut Res, Dept Chem, Ann Arbor, MI 48106 USA
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Parke Davis Pharmaceut Res, Dept Chem, Ann Arbor, MI 48106 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
Metcalf, CA
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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Weigele, M
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0
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ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
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INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
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0
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h-index:
0
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INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
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0
引用数:
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h-index:
0
机构:
INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
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0
引用数:
0
h-index:
0
机构:
INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
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0
引用数:
0
h-index:
0
机构:
INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
Lenoir, C
Dhôtel, H
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0
引用数:
0
h-index:
0
机构:
INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
Dhôtel, H
Garbay, C
论文数:
0
引用数:
0
h-index:
0
机构:
INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
INSERM U266, CNRS FRE 2643, Dept Pharmacochim Mol & Struct, UFR Sci Pharmaceut & Biol, F-75270 Paris 06, France
Garbay, C
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