Novel opioid peptides as kappa opioid receptor antagonists

被引:0
|
作者
Aldrich, JV [1 ]
Wan, Q [1 ]
Murray, TF [1 ]
机构
[1] Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, Baltimore, MD 21201 USA
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:616 / 618
页数:3
相关论文
共 50 条
  • [21] A novel PET radiotracer for imaging the kappa opioid receptor
    Zheng, Ming-Qiang
    Holden, Daniel
    Lin, Shu-Fei
    Mitch, Charlie
    Navarro, Antonio
    Barth, Vanessa
    Quimby, Steve
    Ropchan, Jim
    Carson, Richard E.
    Huang, Yiyun
    JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM, 2012, 32 : S18 - S19
  • [22] A review of the kappa opioid receptor system in opioid use
    Cayir, Salih
    Zhornitsky, Simon
    Barzegary, Alireza
    Sotomayor-Carreno, Esteban
    Sarfo-Ansah, Wonder
    Funaro, Melissa C.
    Matuskey, David
    Angarita, Gustavo
    NEUROSCIENCE AND BIOBEHAVIORAL REVIEWS, 2024, 162
  • [23] Preclinical and clinical efficacy of kappa opioid receptor antagonists for depression: A systematic review
    Wong, Sabrina
    Le, Gia Han
    Vasudeva, Shreya
    Teopiz, Kayla M.
    Phan, Lee
    Meshkat, Shakila
    Kwan, Angela T. H.
    Rhee, Taeho Greg
    Ho, Roger
    Choi, Hayun
    Cao, Bing
    Rosenblat, Joshua D.
    Mcintyre, Roger S.
    JOURNAL OF AFFECTIVE DISORDERS, 2024, 362 : 816 - 827
  • [24] AGONISTS AND ANTAGONISTS BIND TO DIFFERENT DOMAINS OF THE CLONED KAPPA-OPIOID RECEPTOR
    KONG, HY
    RAYNOR, K
    YANO, H
    TAKEDA, J
    BELL, GI
    REISINE, T
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1994, 91 (17) : 8042 - 8046
  • [25] Kappa opioid receptor antagonists: A possible new class of therapeutics for migraine prevention
    Xie, Jennifer Y.
    De Felice, Milena
    Kopruszinski, Caroline M.
    Eyde, Nathan
    LaVigne, Justin
    Remeniuk, Bethany
    Hernandez, Pablo
    Yue, Xu
    Goshima, Naomi
    Ossipov, Michael
    King, Tamara
    Streicher, John M.
    Navratilova, Edita
    Dodick, David
    Rosen, Hugh
    Roberts, Ed
    Porreca, Frank
    CEPHALALGIA, 2017, 37 (08) : 780 - 794
  • [26] Kappa Opioid Receptor Antagonists as Potential Therapeutics for Stress-Related Disorders
    Jacobson, Moriah L.
    Browne, Caroline A.
    Lucki, Irwin
    ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, VOL 60, 2020, 60 : 615 - 636
  • [27] Development of κ Opioid Receptor Antagonists
    Carroll, F. Ivy
    Carlezon, William A., Jr.
    JOURNAL OF MEDICINAL CHEMISTRY, 2013, 56 (06) : 2178 - 2195
  • [28] Transformation of μ-opioid receptor agonists into biologically potent μ-opioid receptor antagonists
    Li, Tingyou
    Jinsmaa, Yunden
    Nedachi, Masahiro
    Miyazaki, Anna
    Tsuda, Yuko
    Ambo, Akihiro
    Sasaki, Yusuke
    Bryant, Sharon D.
    Marczak, Ewa
    Li, Qiang
    Swartzwelder, H. Scott
    Lazarus, Lawrence H.
    Okada, Yoshio
    BIOORGANIC & MEDICINAL CHEMISTRY, 2007, 15 (03) : 1237 - 1251
  • [29] Molecular modeling on kappa opioid receptor and its interaction with nonpeptide kappa opioid agonists
    刘东祥
    蒋华良
    沈敬山
    朱维良
    赵磊
    陈凯先
    嵇汝运
    ActaPharmacologicaSinica, 1999, (02) : 36 - 41
  • [30] Molecular modeling on kappa opioid receptor and its interaction with nonpeptide kappa opioid agonists
    Liu, DX
    Jiang, HL
    Shen, JS
    Zhu, WL
    Zhao, L
    Chen, KX
    Ji, RY
    ACTA PHARMACOLOGICA SINICA, 1999, 20 (02): : 131 - 136