A novel cascade reaction of aryl aldoxime with dimedone under microwave irradiation:: The synthesis of N-hydroxylacridine

被引：94
作者：
Tu, SJ [1 ]
Gao, Y
Fang, F
Zhuang, QY
Feng, YJ
Shi, DQ
机构：
[1] Xuzhou Normal Univ, Key Lab Biotechnol Med Plant, Dept Chem, Xuzhou 221009, Jiangsu, Peoples R China
[2] Shenzhen Univ, Dept Chem, Shenzhen 518060, Guangdong, Peoples R China
来源：
SYNLETT | 2004年 / 02期
关键词：
aryl aldoxime; dimedone; N-hydroxylacridine; micro-wave;
D O I：
10.1055/s-2003-44981
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A novel sequential addition, elimination and cyclization reactions took place when aldoxime and dimedone in glycol was subjected to microwave irradiation and a new type of N-hydroxylacridinedione derivatives was obtained in excellent yields (80-95%) within a short reaction time (4-8 min).
引用
收藏
页码：255 / 258
页数：4
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