Preparation of azaindolines and benzoyl substituted azaindolines: precursors of triazabenzo[cd]azulen-9-one PDE4 inhibitors

被引：8

作者：

Badland, Matthew ^{[1
]}

Devillers, Ingrid ^{[2
]}

Durand, Corinne ^{[2
]}

Fasquelle, Veronique ^{[2
]}

Gaudilliere, Bernard ^{[2
]}

Jacobelli, Henry ^{[2
]}

Manage, Ajith C. ^{[1
]}

Pevet, Isabelle ^{[2
]}

Puaud, Jocelyne ^{[2
]}

Shorter, Anthony J. ^{[1
]}

Wrigglesworth, Roger ^{[2
]}

机构：

[1] Evotec OAI Abingdon, Abingdon OX14 4SD, Oxon, England

[2] Pfizer Global Res & Dev, Fresnes Labs, F-94265 Fresnes, France

来源：

TETRAHEDRON LETTERS | 2011年 / 52卷 / 41期

关键词：

Azaindolines; PDE4; Inhibitors; Pyridine; REVERSE-TRANSCRIPTASE; ANALOGS; PHOSPHODIESTERASE; BROMINATION; NEVIRAPINE; PYRAZINES; PYRIDINES;

D O I：

10.1016/j.tetlet.2011.08.009

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：5292 / 5296

页数：5

共 17 条

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