共 50 条
[31]
Bruton's Tyrosine Kinase Inhibitors: Recent Updates
[J].
Fares, Amneh
;
Uribe, Carlos Carracedo
;
Martinez, Diana
;
Rehman, Tauseef
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Rondon, Carlos Silva
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Sandoval-Sus, Jose
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INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES,
2024, 25 (04)

Fares, Amneh
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Healthcare Syst, Pembroke Pines, FL 33021 USA
Mem Healthcare Syst, Moffitt Malignant Hematol, Pembroke Pines, FL 33021 USA Mem Healthcare Syst, Pembroke Pines, FL 33021 USA

Uribe, Carlos Carracedo
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Healthcare Syst, Pembroke Pines, FL 33021 USA
Mem Healthcare Syst, Moffitt Malignant Hematol, Pembroke Pines, FL 33021 USA Mem Healthcare Syst, Pembroke Pines, FL 33021 USA

Martinez, Diana
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Healthcare Syst, Pembroke Pines, FL 33021 USA
Mem Healthcare Syst, Moffitt Malignant Hematol, Pembroke Pines, FL 33021 USA Mem Healthcare Syst, Pembroke Pines, FL 33021 USA

Rehman, Tauseef
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Healthcare Syst, Pembroke Pines, FL 33021 USA
Mem Healthcare Syst, Moffitt Malignant Hematol, Pembroke Pines, FL 33021 USA Mem Healthcare Syst, Pembroke Pines, FL 33021 USA

Rondon, Carlos Silva
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Healthcare Syst, Moffitt Malignant Hematol, Pembroke Pines, FL 33021 USA Mem Healthcare Syst, Pembroke Pines, FL 33021 USA

Sandoval-Sus, Jose
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Healthcare Syst, Moffitt Malignant Hematol, Pembroke Pines, FL 33021 USA Mem Healthcare Syst, Pembroke Pines, FL 33021 USA
[32]
Cardiovascular Toxicities of Bruton's Tyrosine Kinase Inhibitors
[J].
Pineda-Gayoso, Ricardo
;
Alomar, Mohammed
;
Lee, Dae Hyun
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Fradley, Michael G.
.
CURRENT TREATMENT OPTIONS IN ONCOLOGY,
2020, 21 (08)

Pineda-Gayoso, Ricardo
论文数: 0 引用数: 0
h-index: 0
机构:
Univ S Florida, Div Cardiovasc Med, Morsani Coll Med, Tampa, FL 33620 USA
H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA Univ S Florida, Div Cardiovasc Med, Morsani Coll Med, Tampa, FL 33620 USA

Alomar, Mohammed
论文数: 0 引用数: 0
h-index: 0
机构:
Univ S Florida, Div Cardiovasc Med, Morsani Coll Med, Tampa, FL 33620 USA
H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA Univ S Florida, Div Cardiovasc Med, Morsani Coll Med, Tampa, FL 33620 USA

Lee, Dae Hyun
论文数: 0 引用数: 0
h-index: 0
机构:
Univ S Florida, Div Cardiovasc Med, Morsani Coll Med, Tampa, FL 33620 USA
H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA Univ S Florida, Div Cardiovasc Med, Morsani Coll Med, Tampa, FL 33620 USA

Fradley, Michael G.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Penn, Dept Med, Div Cardiovasc Med, Philadelphia, PA 19104 USA Univ S Florida, Div Cardiovasc Med, Morsani Coll Med, Tampa, FL 33620 USA
[33]
Cardiovascular Toxicities of Bruton’s Tyrosine Kinase Inhibitors
[J].
Ricardo Pineda-Gayoso
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Mohammed Alomar
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Dae Hyun Lee
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Michael G. Fradley
.
Current Treatment Options in Oncology,
2020, 21

Ricardo Pineda-Gayoso
论文数: 0 引用数: 0
h-index: 0
机构: University of South Florida Morsani College of Medicine and H. Lee Moffitt Cancer Center and Research Institute,Division of Cardiovascular Medicine

Mohammed Alomar
论文数: 0 引用数: 0
h-index: 0
机构: University of South Florida Morsani College of Medicine and H. Lee Moffitt Cancer Center and Research Institute,Division of Cardiovascular Medicine

Dae Hyun Lee
论文数: 0 引用数: 0
h-index: 0
机构: University of South Florida Morsani College of Medicine and H. Lee Moffitt Cancer Center and Research Institute,Division of Cardiovascular Medicine

Michael G. Fradley
论文数: 0 引用数: 0
h-index: 0
机构: University of South Florida Morsani College of Medicine and H. Lee Moffitt Cancer Center and Research Institute,Division of Cardiovascular Medicine
[34]
Discovery of Reversible, Noncovalent Bruton's Tyrosine Kinase Inhibitors Targeting BTK C481S Mutation
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Das, Debasis
;
Xie, Lingzhi
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Qiao, Dandan
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Cao, Yuxi
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Jiang, Shanling
;
Zheng, Mei
;
Liu, Zhonghe
;
Li, Yong
;
Jia, Jianhe
;
Lv, Yubin
;
Hong, Jian
.
ACS MEDICINAL CHEMISTRY LETTERS,
2025, 16 (06)
:1038-1047

Das, Debasis
论文数: 0 引用数: 0
h-index: 0
机构:
Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China

Xie, Lingzhi
论文数: 0 引用数: 0
h-index: 0
机构:
Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China

Qiao, Dandan
论文数: 0 引用数: 0
h-index: 0
机构:
Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China

Cao, Yuxi
论文数: 0 引用数: 0
h-index: 0
机构:
Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China

Jiang, Shanling
论文数: 0 引用数: 0
h-index: 0
机构:
Biosun Pharmaceut Co Ltd, Hangzhou 311112, Peoples R China Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China

Zheng, Mei
论文数: 0 引用数: 0
h-index: 0
机构:
Biosun Pharmaceut Co Ltd, Hangzhou 311112, Peoples R China Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China

Liu, Zhonghe
论文数: 0 引用数: 0
h-index: 0
机构:
Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China

Li, Yong
论文数: 0 引用数: 0
h-index: 0
机构:
Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China

Jia, Jianhe
论文数: 0 引用数: 0
h-index: 0
机构:
Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China

Lv, Yubin
论文数: 0 引用数: 0
h-index: 0
机构:
Biosun Pharmaceut Co Ltd, Hangzhou 311112, Peoples R China Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China

Hong, Jian
论文数: 0 引用数: 0
h-index: 0
机构:
Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China Arromax Pharmatech Co Ltd, Suzhou 215123, Peoples R China
[35]
Bruton's Tyrosine Kinase Inhibitors Prevent Therapeutic Escape in Breast Cancer Cells
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Wang, Xianhui
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Wong, Jason
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Sevinsky, Christopher J.
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Kokabee, Leila
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Khan, Faiza
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Sun, Yan
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Conklin, Douglas S.
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MOLECULAR CANCER THERAPEUTICS,
2016, 15 (09)
:2198-2208

Wang, Xianhui
论文数: 0 引用数: 0
h-index: 0
机构:
SUNY Albany, Canc Res Ctr, Rensselaer, NY USA
SUNY Albany, Dept Biomed Sci, Rensselaer, NY USA SUNY Albany, Canc Res Ctr, Rensselaer, NY USA

Wong, Jason
论文数: 0 引用数: 0
h-index: 0
机构:
SUNY Albany, Canc Res Ctr, Rensselaer, NY USA
SUNY Albany, Dept Biomed Sci, Rensselaer, NY USA SUNY Albany, Canc Res Ctr, Rensselaer, NY USA

Sevinsky, Christopher J.
论文数: 0 引用数: 0
h-index: 0
机构:
SUNY Albany, Canc Res Ctr, Rensselaer, NY USA
SUNY Albany, Dept Biomed Sci, Rensselaer, NY USA SUNY Albany, Canc Res Ctr, Rensselaer, NY USA

Kokabee, Leila
论文数: 0 引用数: 0
h-index: 0
机构:
SUNY Albany, Canc Res Ctr, Rensselaer, NY USA
SUNY Albany, Dept Biomed Sci, Rensselaer, NY USA
Pasteur Inst Iran, Dept Mol Med, Tehran, Iran SUNY Albany, Canc Res Ctr, Rensselaer, NY USA

Khan, Faiza
论文数: 0 引用数: 0
h-index: 0
机构:
SUNY Albany, Canc Res Ctr, Rensselaer, NY USA
SUNY Albany, Dept Biomed Sci, Rensselaer, NY USA SUNY Albany, Canc Res Ctr, Rensselaer, NY USA

Sun, Yan
论文数: 0 引用数: 0
h-index: 0
机构:
SUNY Albany, Canc Res Ctr, Rensselaer, NY USA
SUNY Albany, Dept Biomed Sci, Rensselaer, NY USA SUNY Albany, Canc Res Ctr, Rensselaer, NY USA

Conklin, Douglas S.
论文数: 0 引用数: 0
h-index: 0
机构:
SUNY Albany, Canc Res Ctr, Rensselaer, NY USA
SUNY Albany, Dept Biomed Sci, Rensselaer, NY USA SUNY Albany, Canc Res Ctr, Rensselaer, NY USA
[36]
Bayesian machine learning to discover Bruton's tyrosine kinase inhibitors
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Wang, Jian
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Ran, Ting
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Chen, Yadong
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Lu, Tao
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CHEMICAL BIOLOGY & DRUG DESIGN,
2020, 96 (04)
:1113-1121

Wang, Jian
论文数: 0 引用数: 0
h-index: 0
机构:
China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China
Zhejiang Pharmaceut Coll, Ningbo, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China

Ran, Ting
论文数: 0 引用数: 0
h-index: 0
机构:
Xiamen Univ, Sch Pharmaceut Sci, Fujian Prov Key Lab Innovat Drug Target Res, Xiamen, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China

Chen, Yadong
论文数: 0 引用数: 0
h-index: 0
机构:
China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China

Lu, Tao
论文数: 0 引用数: 0
h-index: 0
机构:
China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China
[37]
Design and discovery of new selective and potent VEGF receptor 2 tyrosine kinase inhibitors
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Hou, Fei
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Yao, Yuhong
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Wei, Yujiao
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Wang, Yubo
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Cao, Yangzi
;
Liu, Xinqiang
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Zheng, Liting
;
Zhang, Qingqing
;
Jiao, Yue
;
Chen, Yukun
;
Meng, Yue
;
Sun, Yue
;
Wu, Yanjie
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Wang, Jiefu
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Wang, Junfeng
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Wu, Zhou
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Zhang, Kun
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Wei, Mingming
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Yang, Guang
.
BIOORGANIC & MEDICINAL CHEMISTRY,
2023, 91

Hou, Fei
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Yao, Yuhong
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Wei, Yujiao
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Wang, Yubo
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Cao, Yangzi
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Liu, Xinqiang
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Zheng, Liting
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Zhang, Qingqing
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Jiao, Yue
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Chen, Yukun
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Meng, Yue
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Sun, Yue
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Wu, Yanjie
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Wang, Jiefu
论文数: 0 引用数: 0
h-index: 0
机构:
Tianjin Med Univ Canc Inst & Hosp, Natl Clin Res Ctr Canc, Tianjins Clin Res Ctr Canc, Key Lab Canc Prevent & Therapy, Tianjin 300060, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Wang, Junfeng
论文数: 0 引用数: 0
h-index: 0
机构:
Tianjin Med Univ Canc Inst & Hosp, Natl Clin Res Ctr Canc, Tianjins Clin Res Ctr Canc, Key Lab Canc Prevent & Therapy, Tianjin 300060, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Wu, Zhou
论文数: 0 引用数: 0
h-index: 0
机构:
China Resources Biopharmaceut Co Ltd, Beijing 100100, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Zhang, Kun
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Wei, Mingming
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China

Yang, Guang
论文数: 0 引用数: 0
h-index: 0
机构:
Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China Nankai Univ, Coll Life Sci, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China
[38]
Bruton's Tyrosine Kinase Inhibitors in Chronic Lymphocytic Leukemia and Lymphoma
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Varma, Gaurav
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Johnson, Tyler P.
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Advani, Ranjana H.
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CLINICAL ADVANCES IN HEMATOLOGY & ONCOLOGY,
2016, 14 (07)
:543-554

论文数: 引用数:
h-index:
机构:

Johnson, Tyler P.
论文数: 0 引用数: 0
h-index: 0
机构:
Stanford Univ, Med Ctr, Dept Med, Div Oncol, Stanford, CA 94305 USA Drexel Univ, Coll Med, Philadelphia, PA 19104 USA

Advani, Ranjana H.
论文数: 0 引用数: 0
h-index: 0
机构:
Stanford Univ, Med Ctr, Dept Med, Div Oncol,Lymphoma, Stanford, CA 94305 USA
Stanford Univ, Med Ctr, Dept Med, Div Oncol,Med & Oncol, Stanford, CA 94305 USA Drexel Univ, Coll Med, Philadelphia, PA 19104 USA
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Selective Inhibition of Bruton?s Tyrosine Kinase by a Designed Covalent Ligand Leads to Potent Therapeutic Efficacy in Blood Cancers Relative to Clinically Used Inhibitors
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Sousa, Barbara B.
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De Almeida, Catia Rebelo
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Barahona, Ana F.
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Lopes, Raquel
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Martins-Logrado, Ana
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Cavaco, Marco
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Neves, Vera
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Carvalho, Luis A. R.
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Labao-Almeida, Carlos
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Coelho, Ana R.
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Bento, Marta Leal
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Lopes, Ricardo M. R. M.
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Oliveira, Bruno L.
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Castanho, Miguel A. R. B.
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Neumeister, Peter
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Deutsch, Alexander
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Vladimer, Gregory I.
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Krall, Nikolaus
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Joao, Cristina
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Corzana, Francisco
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Seixas, Joao D.
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Fior, Rita
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Bernardes, Goncalo J. L.
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ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE,
2022, 5 (11)
:1156-1168

Sousa, Barbara B.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

De Almeida, Catia Rebelo
论文数: 0 引用数: 0
h-index: 0
机构:
Champalimaud Fdn, P-1400038 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Barahona, Ana F.
论文数: 0 引用数: 0
h-index: 0
机构:
Champalimaud Fdn, P-1400038 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Lopes, Raquel
论文数: 0 引用数: 0
h-index: 0
机构:
Champalimaud Fdn, P-1400038 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Martins-Logrado, Ana
论文数: 0 引用数: 0
h-index: 0
机构:
Champalimaud Fdn, P-1400038 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Cavaco, Marco
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Neves, Vera
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Carvalho, Luis A. R.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Cambridge, Yusuf Hamied Dept Chem, Cambridge CB2 1EW, England Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Labao-Almeida, Carlos
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Coelho, Ana R.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Bento, Marta Leal
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal
Ctr Hospitalar Lisboa Norte, Dept Hematol & Bone Marrow Transplantat, P-1649035 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Lopes, Ricardo M. R. M.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Lisbon, Res Inst Med iMed ULisboa, Fac Farm, P-1600277 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Oliveira, Bruno L.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Castanho, Miguel A. R. B.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Neumeister, Peter
论文数: 0 引用数: 0
h-index: 0
机构:
Med Univ Graz, Div Hematol, A-8036 Graz, Austria Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

论文数: 引用数:
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Vladimer, Gregory I.
论文数: 0 引用数: 0
h-index: 0
机构:
Exscientia, Oxford OX4 4GE, England Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Krall, Nikolaus
论文数: 0 引用数: 0
h-index: 0
机构:
Exscientia, Oxford OX4 4GE, England Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Joao, Cristina
论文数: 0 引用数: 0
h-index: 0
机构:
Champalimaud Fdn, P-1400038 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Corzana, Francisco
论文数: 0 引用数: 0
h-index: 0
机构:
Univ La Rioja, Ctr Invest Sintesis Quim, Dept Quim, Logrono 26006, Spain Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Seixas, Joao D.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal
TARGTEX SA, Torres Vedras P-2560275, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Fior, Rita
论文数: 0 引用数: 0
h-index: 0
机构:
Champalimaud Fdn, P-1400038 Lisbon, Portugal Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal

Bernardes, Goncalo J. L.
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机构:
Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal
Univ Cambridge, Yusuf Hamied Dept Chem, Cambridge CB2 1EW, England Univ Lisbon, Fac Med, Inst Med Mol Joao Lobo Antunes, P-1649028 Lisbon, Portugal
[40]
Discovery of BIIB068: A Selective, Potent, Reversible Bruton's Tyrosine Kinase Inhibitor as an Orally Efficacious Agent for Autoimmune Diseases
[J].
Ma, Bin
;
Bohnert, Tonika
;
Otipoby, Kevin L.
;
Tien, Eric
;
Arefayene, Million
;
Bai, Judy
;
Bajrami, Bekim
;
Bame, Eris
;
Chan, Timothy R.
;
Humora, Michael
;
MacPhee, J. Michael
;
Marcotte, Douglas
;
Mehta, Devangi
;
Metrick, Claire M.
;
Moniz, George
;
Polack, Evelyne
;
Poreci, Urjana
;
Prefontaine, Annick
;
Sheikh, Sarah
;
Schroeder, Patricia
;
Smirnakis, Karen
;
Zhang, Lei
;
Zheng, Fengmei
;
Hopkins, Brian T.
.
JOURNAL OF MEDICINAL CHEMISTRY,
2020, 63 (21)
:12526-12541

Ma, Bin
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机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Bohnert, Tonika
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Otipoby, Kevin L.
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Tien, Eric
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Arefayene, Million
论文数: 0 引用数: 0
h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Bai, Judy
论文数: 0 引用数: 0
h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Bajrami, Bekim
论文数: 0 引用数: 0
h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Bame, Eris
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Chan, Timothy R.
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Humora, Michael
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

MacPhee, J. Michael
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Marcotte, Douglas
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Mehta, Devangi
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Metrick, Claire M.
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Moniz, George
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机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Polack, Evelyne
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机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Poreci, Urjana
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Prefontaine, Annick
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Sheikh, Sarah
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Schroeder, Patricia
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h-index: 0
机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Smirnakis, Karen
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机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Zhang, Lei
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机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Zheng, Fengmei
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机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA

Hopkins, Brian T.
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机构:
Biogen, Res & Dev, Cambridge, MA 02142 USA Biogen, Res & Dev, Cambridge, MA 02142 USA