Synthesis of Stable σ-Adducts by Arylation of Quinazoline

被引:1
作者
Azev, Yu. A. [1 ]
Koptyaeva, O. S. [1 ]
Seliverstova, E. A. [1 ]
Ivoilova, A. V. [1 ]
Pospelova, T. A. [1 ]
机构
[1] Yeltsin Ural Fed Univ, Ekaterinburg, Russia
基金
俄罗斯基础研究基金会;
关键词
quinazoline; C-nucleophiles; C-C-bond formation; DERIVATIVES;
D O I
10.1134/S1070363219120089
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
The reactions of quinazoline with 1,3,5-trimethoxybenzene, 3- and 4-methylbenzene-1,2-diamines, and 1-(4-methoxybenzylidene)-2-phenylhydrazine on heating in the presence of trifluoroacetic acid afforded the corresponding stable C-C sigma-adducts.
引用
收藏
页码:2374 / 2377
页数:4
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