FeCl3 AND MORPHOLINE AS EFFICIENT COCATALYSTS FOR THE ONE-STEP SYNTHESIS OF QUINOXALINES FROM α-HYDROXYKETONES AND 1,2-DIAMINES

被引:26
作者
Song, Weibin [1 ]
Liu, Peng [1 ]
Lei, Min [1 ]
You, Hanyun [1 ]
Chen, Xubing [1 ]
Chen, Hu [1 ]
Ma, Lei [1 ]
Hu, Lihong [1 ,2 ]
机构
[1] E China Univ Sci & Technol, Sch Pharm, Shanghai 200237, Peoples R China
[2] Chinese Acad Sci, Shanghai Inst Mat Med, Shanghai 200031, Peoples R China
基金
中国国家自然科学基金;
关键词
Cocatalyst; FeCl3; morpholine; quinoxaline; OXIDATION PROCESSES; CATALYZED SYNTHESIS; AMMONIUM-NITRATE; IRON COMPLEX; DERIVATIVES; SOLVENT; GREEN; ACID; CYCLIZATION; CONVENIENT;
D O I
10.1080/00397911.2010.523489
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
One-step conversion including intramolecular hydrogen bond decomposition, aerobic oxidation, and condensation from alpha-hydroxyketones and 1,2-diamines into quinoxalines is reported using FeCl3 and morpholine as cocatalysts.
引用
收藏
页码:236 / 245
页数:10
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