Molecular diversity of four-component synthesis of pyrazole-based pyrido[2,3-d]pyrimidine-diones in water: a green synthesis

被引：12
作者：
Daraie, Mansoureh [1 ]
Heravi, Majid M. [1 ]
机构：
[1] Alzahra Univ, Sch Sci, Dept Chem, Tehran, Iran
来源：
ARKIVOC | 2016年
关键词：
Pyrazole; pyrido[2,3-d]pyrimidine-diones; green synthesis; four-component reaction; ONE-POT SYNTHESIS; MULTICOMPONENT REACTIONS; REGIOSELECTIVE SYNTHESIS; EFFICIENT CATALYST; TUBERCULOSIS; DERIVATIVES;
D O I：
10.3998/ark.5550190.p009.603
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A novel one pot, four component synthesis of pyrazolo[4',3':5,6]pyrido[2,3-d]pyrimidine-diones, involving, hydrazine hydrate, ethyl acetoacetate, 6-amino-1,3-dimethyl uracil and an appropriate aryl aldehyde in the presence of two green catalysts in water, is reported.
引用
收藏
页码：328 / 338
页数：11
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