共 34 条
Rituximab (anti-CD20)-modified AZD-2014-encapsulated nanoparticles killing of B lymphoma cells
被引:9
作者:

Tang, Xiaolong
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Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China

Xie, Chunmei
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h-index: 0
机构:
Guangzhou Med Univ, Guangzhou Peoples Hosp 8, Dept Lab Med, Guangzhou, Guangdong, Peoples R China Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China

Jiang, Zhenyou
论文数: 0 引用数: 0
h-index: 0
机构:
Jinan Univ, Dept Microbiol, Guangzhou, Guangdong, Peoples R China
Jinan Univ, Dept Immunol, Guangzhou, Guangdong, Peoples R China Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China

Li, Amin
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h-index: 0
机构:
Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China

Cai, Shiyu
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Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China

Hou, Changhao
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h-index: 0
机构:
Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China

Wang, Jian
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h-index: 0
机构:
Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China

Liang, Yong
论文数: 0 引用数: 0
h-index: 0
机构:
Xuzhou Med Coll, Huaian Hosp, Huaian, Peoples R China
Huaian Second Hosp, Huaian, Peoples R China Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China

Ma, Dong
论文数: 0 引用数: 0
h-index: 0
机构:
Jinan Univ, Dept Biomed Engn, Guangdong Higher Educ Inst, Key Lab Biomat, Guangzhou, Guangdong, Peoples R China Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China
机构:
[1] Anhui Univ Sci & Technol, Med Coll, Huainan, Peoples R China
[2] Guangzhou Med Univ, Guangzhou Peoples Hosp 8, Dept Lab Med, Guangzhou, Guangdong, Peoples R China
[3] Jinan Univ, Dept Microbiol, Guangzhou, Guangdong, Peoples R China
[4] Jinan Univ, Dept Immunol, Guangzhou, Guangdong, Peoples R China
[5] Xuzhou Med Coll, Huaian Hosp, Huaian, Peoples R China
[6] Huaian Second Hosp, Huaian, Peoples R China
[7] Jinan Univ, Dept Biomed Engn, Guangdong Higher Educ Inst, Key Lab Biomat, Guangzhou, Guangdong, Peoples R China
基金:
中国国家自然科学基金;
关键词:
Non-Hodgkin's lymphoma;
mTOR;
signal pathways;
rituximab;
nanoparticles;
TOR serine-threonine kinases;
AZD-2014;
NON-HODGKINS-LYMPHOMA;
PRECLINICAL EVALUATION;
INHIBITOR;
MTOR;
METABOLISM;
ACTIVATION;
INITIATION;
APOPTOSIS;
PATHWAYS;
GROWTH;
D O I:
10.1080/21691401.2018.1478844
中图分类号:
Q81 [生物工程学(生物技术)];
Q93 [微生物学];
学科分类号:
071005 ;
0836 ;
090102 ;
100705 ;
摘要:
The mTOR signal pathway is often highly activated in B-cell non-Hodgkin's lymphoma (NHL) and promotes cancer progression and chemo-resistance. Therefore, the pathways of mTOR are an important target for drug development in this disease. In the current study, we developed a rituximab (anti-CD20)-modified mTOR inhibitor, AZD-2014, loaded into nanoparticles (Ab-NPs-AZD-2014) for trial of its anti-NHL effect. In a cultured NHL cell line, Ab-NPs-AZD-2014 inhibited cancer cell growth, induced cell apoptosis, and blocked activation of mTORC1 and mTORC2 in Raji cells. These results indicate that antibody modification and nanomaterial loading of AZD-2014 with anti-CD20 significantly improved efficacy of AZD-2014 against NHL cells. This approach may ultimately deserve testing in therapy against NHL.
引用
收藏
页码:1063 / 1073
页数:11
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