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- [1] Discovery of selective orexin-1 receptor antagonistsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 254Shireman, Brock论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USAPreville, Cathy论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USAZiff, Jeannie论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USADvorak, Curt论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USACoate, Heather论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USAGelin, Christine论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USALebold, Terry论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USABonaventure, Pascal论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USADugovic, Christine论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USAKoudriakova, Tatiana论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USALord, Brian论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USANepomuceno, Diane论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USAShelton, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USALovenberg, Timothy论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USACarruthers, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, San Diego, CA USA Janssen Pharmaceut Res & Dev, San Diego, CA USA
- [2] Selective orexin receptor antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (17) : 4761 - 4769Lebold, Terry P.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, San Diego, CA 92121 USA Janssen Res & Dev, San Diego, CA 92121 USABonaventure, Pascal论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, San Diego, CA 92121 USA Janssen Res & Dev, San Diego, CA 92121 USAShireman, Brock T.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, San Diego, CA 92121 USA Janssen Res & Dev, San Diego, CA 92121 USA
- [3] Discovery of piperidine ethers as selective orexin receptor antagonists (SORAs) inspired by filorexantBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 25 (03) : 444 - 450Raheem, Izzat T.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USABreslin, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USABruno, Joseph论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USACabalu, Tamara D.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Pharmacokinet Pharmacodynam & Drug Metab, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USACooke, Andrew论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USACox, Christopher D.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USACui, Donghui论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Pharmacokinet Pharmacodynam & Drug Metab, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USAGarson, Susan论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USAGotter, Anthony L.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USAFox, Steven V.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Vivo Pharmacol, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USAHarrell, C. Meacham论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USAKuduk, Scott D.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USALemaire, Wei论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Vitro Pharmacol, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USAPrueksaritanont, Thomayant论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Pharmacokinet Pharmacodynam & Drug Metab, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USARenger, John J.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USAStump, Craig论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USATannenbaum, Pamela L.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Vivo Pharmacol, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USAWilliams, Peter D.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USAWinrow, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USAColeman, Paul J.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Discovery Chem, West Point, PA 19486 USA
- [4] PHARMACOLOGICAL CHARACTERIZATION OF OREXIN RECEPTOR ANTAGONISTSSLEEP, 2011, 34 : A5 - A5Winrow, C. J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USADoran, S. M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USAGotter, A. L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USAPausch, M. H.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USAKuduk, S. D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USAUslaner, J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USACarroll, S. S.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USASmith, S.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USAColeman, P. J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USARenger, J. J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USA
- [5] Discovery of spiropiperidine-based potent and selective Orexin-2 receptor antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (21) : 6409 - 6413Fujimoto, Tatsuhiko论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co, Med Chem Res Labs, Kanagawa 2511238, Japan Takeda Pharmaceut Co, Med Chem Res Labs, Kanagawa 2511238, JapanTomata, Yoshihide论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co, Med Chem Res Labs, Kanagawa 2511238, Japan Takeda Pharmaceut Co, Med Chem Res Labs, Kanagawa 2511238, JapanKunitomo, Jun论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co, Med Chem Res Labs, Kanagawa 2511238, Japan Takeda Pharmaceut Co, Med Chem Res Labs, Kanagawa 2511238, JapanHirozane, Mariko论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co, Discovery Res Labs, Kanagawa 2511238, Japan Takeda Pharmaceut Co, Med Chem Res Labs, Kanagawa 2511238, JapanMarui, Shogo论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co, Med Chem Res Labs, Kanagawa 2511238, Japan Takeda Pharmaceut Co, Med Chem Res Labs, Kanagawa 2511238, Japan
- [6] Discovery and development of orexin receptor antagonists as therapeutics for insomniaBRITISH JOURNAL OF PHARMACOLOGY, 2014, 171 (02) : 283 - 293Winrow, C. J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, West Point, PA USA Merck Res Labs, Dept Neurosci, West Point, PA USARenger, J. J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, West Point, PA USA Merck Res Labs, Dept Neurosci, West Point, PA USA
- [7] Investigation of orexin-2 selective receptor antagonists: Structural modifications resulting in dual orexin receptor antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 27 (06) : 1364 - 1370Skudlarek, Jason W.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USADiMarco, Christina N.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USABabaoglu, Kerim论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Chem Capabil & Screening, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USARoecker, Anthony J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USABruno, Joseph G.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Vitro Pharmacol, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USAPausch, Mark A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Vitro Pharmacol, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USAO'Brien, Julie A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Vitro Pharmacol, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USACabalu, Tamara D.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Drug Metab, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USAStevens, Joanne论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Vivo Pharmacol, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USABrunner, Joseph论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Neurosci, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USATannenbaum, Pamela L.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Vivo Pharmacol, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USAWuelfing, W. Peter论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Discovery Pharmaceut Sci, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USAGarson, Susan L.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Neurosci, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USAFox, Steven V.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Vivo Pharmacol, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USASavitz, Alan T.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Vivo Pharmacol, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USAHarrell, Charles M.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Neurosci, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USAGotter, Anthony L.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Neurosci, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USAWinrow, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Neurosci, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USARenger, John J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Neurosci, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USAKuduk, Scott D.论文数: 0 引用数: 0 h-index: 0机构: Novira Therapeut Inc, Janssen Pharmaceut, Doylestown, PA 18902 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USAColeman, Paul J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USA Merck & Co Inc, MRL, Dept Med Chem, West Point, PA 19486 USA
- [8] Selective orexin receptor antagonists for the treatment of CNS disordersABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2013, 245Shireman, Brock T.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USALetavic, Michael A.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USABonaventure, Pascal论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USABranstetter, Bryan论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USADugovic, Christine论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USAHack, Michael论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USALord, Brian论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USALy, Kiev S.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USAMorton, Kirsten L.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USARudolph, Dale A.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USASavall, Brad M.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USAShah, Chandra论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USAShelton, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USAShoblock, James论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USANepomuceno, Diane论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USALovenberg, Timothy W.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USACarruthers, Nicholas I.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA Janssen Res & Dev LLC, Dept Neurosci, San Diego, CA 92121 USA
- [9] Substituted Tetrahydroisoquinolines as Selective Antagonists for the Orexin 1 ReceptorJOURNAL OF MEDICINAL CHEMISTRY, 2013, 56 (17) : 6901 - 6916Perrey, David A.论文数: 0 引用数: 0 h-index: 0机构: Res Triangle Inst, Res Triangle Pk, NC 27709 USA Res Triangle Inst, Res Triangle Pk, NC 27709 USAGerman, Nadezhda A.论文数: 0 引用数: 0 h-index: 0机构: Res Triangle Inst, Res Triangle Pk, NC 27709 USA Res Triangle Inst, Res Triangle Pk, NC 27709 USAGilmour, Brian P.论文数: 0 引用数: 0 h-index: 0机构: Res Triangle Inst, Res Triangle Pk, NC 27709 USA Res Triangle Inst, Res Triangle Pk, NC 27709 USALi, Jun-Xu论文数: 0 引用数: 0 h-index: 0机构: SUNY Buffalo, Dept Pharmacol & Toxicol, Buffalo, NY 14214 USA Res Triangle Inst, Res Triangle Pk, NC 27709 USAHarris, Danni L.论文数: 0 引用数: 0 h-index: 0机构: Res Triangle Inst, Res Triangle Pk, NC 27709 USA Res Triangle Inst, Res Triangle Pk, NC 27709 USAThomas, Brian F.论文数: 0 引用数: 0 h-index: 0机构: Res Triangle Inst, Res Triangle Pk, NC 27709 USA Res Triangle Inst, Res Triangle Pk, NC 27709 USAZhang, Yanan论文数: 0 引用数: 0 h-index: 0机构: Res Triangle Inst, Res Triangle Pk, NC 27709 USA Res Triangle Inst, Res Triangle Pk, NC 27709 USA
- [10] Discovery of highly potent and selective orexin 1 receptor antagonists (1-SORAs) suitable for in vivo interrogation of orexin 1 receptor pharmacologyBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 26 (23) : 5809 - 5814Stump, Craig A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USACooke, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USABruno, Joseph论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Vitro Pharmacol, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USACabalu, Tamara D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Pharmacokinet Pharmacodynam & Drug Metab, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAGotter, Anthony L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurosci, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAHarell, C. Meacham论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurosci, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAKuduk, Scott D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAMcDonald, Terrence P.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurosci, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAO'Brien, Julie论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Vitro Pharmacol, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USARenger, John J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurosci, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAWilliams, Peter D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAWinrow, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurosci, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAColeman, Paul J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USA