Development of a large-scale synthesis of denagliptin tosylate

被引:0
作者
Powers, Jeremiah [1 ]
机构
[1] GlaxoSmithKline Inc, Dept API Chem & Anal, Res Triangle Pk, NC 27709 USA
来源
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2011年 / 242卷
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
550-ORGN
引用
收藏
页数:1
相关论文
共 50 条
[41]   Development of a Large-Scale Route to Glecaprevir: Synthesis of the Side Chain and Final Assembly [J].
Hill, David R. ;
Abrahamson, Michael J. ;
Lukin, Kirill A. ;
Towne, Timothy B. ;
Engstrom, Kenneth M. ;
Reddy, Rajarathnam E. ;
Kielbus, Angelica B. ;
Pelc, Matthew J. ;
Mei, Jianzhang ;
Nere, Nandkishor K. ;
Chen, Shuang ;
Henry, Rodger ;
Chemburkar, Sanjay ;
Ding, Chen ;
Zhang, Hongqiang ;
Cink, Russell D. .
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2020, 24 (08) :1393-1404
[42]   Synthesis and Development of a Nonaflate Ester in the Large-Scale Preparation of 3-Deoxymorphine [J].
Ruda, Antonio M. ;
Moseley, Jonathan D. .
LETTERS IN ORGANIC CHEMISTRY, 2024, 21 (09) :744-748
[43]   Development of a Fit-for-Purpose Large-Scale Synthesis of an Oral PARP Inhibitor [J].
Wallace, Debra J. ;
Baxter, Carl A. ;
Brands, Karel J. M. ;
Bremeyer, Nadine ;
Brewer, Sarah E. ;
Desmond, Richard ;
Emerson, Khateeta M. ;
Foley, Jennifer ;
Fernandez, Paul ;
Hu, Weifeng ;
Keen, Stephen P. ;
Mullens, Peter ;
Muzzio, Daniel ;
Sajonz, Peter ;
Tan, Lushi ;
Wilson, Robert D. ;
Zhou, George ;
Zhou, Guoyue .
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2011, 15 (04) :831-840
[44]   Large-scale synthesis and forming of xerogel catalysts [J].
Alie, C. ;
Ferauche, F. ;
Tcherkassova, N. ;
Pirard, R. ;
Lambert, S. ;
Winterton, N. ;
Pirard, J. -P. ;
Heinrichs, B. .
SCIENTIFIC BASES FOR THE PREPARATION OF HETEROGENEOUS CATALYSTS, PROCEEDINGS OF THE 9TH INTERNATIONAL SYMPOSIUM, 2006, 162 :729-736
[45]   LARGE-SCALE SYNTHESIS OF DIAMMONIUM ACETYL PHOSPHATE [J].
WHITESIDES, GM ;
SIEGEL, M ;
GARRETT, P .
JOURNAL OF ORGANIC CHEMISTRY, 1975, 40 (17) :2516-2519
[46]   LARGE-SCALE SYNTHESIS OF ANTISENSE OLIGODEOXYRIBONUCLEOTIDE PHOSPHOROTHIOATE [J].
TANG, JX ;
TANG, JY .
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1995, 209 :222-MEDI
[47]   Synthesis of Large-Scale Instant IoT Networks [J].
Ghosh, Pradipta ;
Bunton, Jonathan ;
Pylorof, Dimitrios ;
Vieira, Marcos A. M. ;
Chan, Kevin ;
Govindan, Ramesh ;
Sukhatme, Gaurav S. S. ;
Tabuada, Paulo ;
Verma, Gunjan .
IEEE TRANSACTIONS ON MOBILE COMPUTING, 2023, 22 (03) :1810-1824
[48]   Large-scale synthesis of glycoconjugates through biotechnology [J].
Wang, PG .
GLYCOBIOLOGY, 2001, 11 (10) :934-934
[49]   Large-scale green synthesis of Cu nanoparticles [J].
A. B. S. Sastry ;
R. B. Karthik Aamanchi ;
Ch. Sree Rama Linga Prasad ;
B. S. Murty .
Environmental Chemistry Letters, 2013, 11 :183-187
[50]   AN IMPROVED, LARGE-SCALE SYNTHESIS OF XANTHOTHRICIN AND REUMYCIN [J].
BLACK, TH .
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1987, 24 (05) :1373-1375