Synthesis of biheterocyclic α-aminophosphonic acid derivatives

被引：6

作者：

Achamlale, S

Elachqar, A

El Hallaoui, A

Alami, A

Elhajji, S

Roumestant, ML

Viallefont, P

机构：

[1] Univ Montpellier 2, Chim Organ Lab, UMR 5810, F-34060 Montpellier, France

[2] Univ Sidi Mohamed Ben Abdellah, Fac Sci Dhar El Mehraz, Chim Organ Lab, Fes, Morocco

来源：

PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS | 1998年 / 140卷

关键词：

alpha-aminophosphonic acid; biheterocycle; 1,2,3-triazole; tetrazole;

D O I：

10.1080/10426509808035736

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

We report here the synthesis of biheterocyclic alpha -aminophosphonic acid derivatives by 1,3 dipolar cycloaddition of acetylenic compounds, prepared in the laboratory, on alpha -azido alpha -amino phosphonic esters 1([1a]).

引用

页码：103 / 111

页数：9

共 17 条

[1] Synthesis of alpha-triazolyl alpha-amino acid derivatives [J].

Achamlal, S ;

Elachqar, A ;

ElHallaoui, A ;

ElHajji, S ;

Roumestant, ML ;

Viallefont, P .

AMINO ACIDS, 1997, 12 (3-4) :257-263

[2]

ACHAMLALE S, IN PRESS J HETEROCYC

[3]

Alami A, 1996, B SOC CHIM BELG, V105, P769

[4]

ANTONOWA A, 1976, Z CHEM, V16, P17

[5] FROM OXAZOLINES TO PRECURSORS OF AMINO-ACIDS [J].

ATMANI, A ;

ELHALLAOUI, A ;

ELHAJJI, S ;

ROUMESTANT, ML ;

VIALLEFONT, P .

SYNTHETIC COMMUNICATIONS, 1991, 21 (22) :2383-2390

[6] C-13-H COUPLING-CONSTANTS AS A TOOL IN TAUTOMERISM STUDIES OF 1,2,3-TRIAZOLE, 1,2,4-TRIAZOLE, AND TETRAZOLE [J].

BEGTRUP, M .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 2, 1976, (06) :736-741

[7] SUBSTITUTIONS- UND ADDITIONSREAKTIONEN AN SILYLIERTEN ACETYLENEN [J].

BIRKOFER, L ;

UHLENBRA.H ;

RITTER, A .

CHEMISCHE BERICHTE-RECUEIL, 1963, 96 (12) :3280-&

[8] SYNTHESIS OF HETEROCYCLIC ALPHA-AMINOPHOSPHONIC ACIDS [J].

ELACHQAR, A ;

ELHALLAOUI, A ;

ROUMESTANT, ML ;

VIALLEFONT, P .

SYNTHETIC COMMUNICATIONS, 1994, 24 (09) :1279-1286

[9] C-13 MAGNETIC-RESONANCE STUDIES OF AZOLES - TAUTOMERISM, SHIFT-REAGENT EFFECTS, AND SOLVENT EFFECTS [J].

ELGUERO, J ;

MARZIN, C ;

ROBERTS, JD .

JOURNAL OF ORGANIC CHEMISTRY, 1974, 39 (03) :357-363

[10] BIOLOGICAL-ACTIVITY OF AMINOPHOSPHONIC ACIDS [J].

KAFARSKI, P ;

LEJCZAK, B .

PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 1991, 63 (1-2) :193-215

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