A Review on Domino Condensation/Cyclization Reactions for the Synthesis of 2-Substituted 1,3-Benzothiazole Derivatives

被引：66
|
作者：
Liu, Xing [1 ]
Dong, Zhi-Bing [1 ,2 ,3 ,4 ]
机构：
[1] Wuhan Inst Technol, Sch Chem & Environm Engn, Wuhan 430205, Peoples R China
[2] Wuhan Inst Technol, Minist Educ, Key Lab Green Chem Proc, Minist Educ, Wuhan 430205, Peoples R China
[3] Hubei Univ, Minist Educ, Key Lab Synth & Applicat Organ Funct Mol, Wuhan 430062, Peoples R China
[4] Wuhan Inst Technol, Hubei Key Lab Novel Reactor & Green Chem Technol, Wuhan 430205, Peoples R China
来源：
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY | 2020年 / 2020卷 / 04期
基金：
中国国家自然科学基金;
关键词：
Benzothiazoles; Cyclization; Condensation; Heterocycles; Synthetic methods; ONE-POT SYNTHESIS; HIGHLY EFFICIENT SYNTHESIS; CATALYZED S-ARYLATION; SOLVENT-FREE; BENZOTHIAZOLE DERIVATIVES; FACILE SYNTHESIS; ENVIRONMENTALLY BENIGN; HETEROCYCLIC THIONES; TANDEM REACTION; GREEN SYNTHESIS;
D O I：
10.1002/ejoc.201901502
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Domino reactions serve as one of the most step-economical methods for the synthesis of benzoxazole molecules such as 2-substituted 1,3-benzothiazoles. Recently, a variety of compounds were found to facilitate these domino reactions. Here, we have summarized the most important domino condensation and cyclization reactions in view of the formation of 2-substituted 1,3-benzothiazoles using specific cyclization agents.
引用
收藏
页码：408 / 419
页数：12
相关论文
共 50 条
  • [1] Synthesis and Biological Activity of New 1,3-Benzothiazole Derivatives
    N. A. Pulina
    F. V. Sobin
    T. A. Yushkova
    T. F. Odegova
    A. I. Krasnova
    Pharmaceutical Chemistry Journal, 2014, 48 : 505 - 508
  • [2] Synthesis and Biological Activity of New 1,3-Benzothiazole Derivatives
    Pulina, N. A.
    Sobin, F. V.
    Yushkova, T. A.
    Odegova, T. F.
    Krasnova, A. I.
    PHARMACEUTICAL CHEMISTRY JOURNAL, 2014, 48 (08) : 505 - 508
  • [3] The nitration and bromination of 2-(pentafluorosulfanyl)-1,3-benzothiazole and 2-(trifluoromethyl)-1,3-benzothiazole
    Olexandr I. Guzyr
    Lyudmila M. Potikha
    Svitlana V. Shishkina
    Volodymyr N. Fetyukhin
    Yuriy G. Shermolovich
    Chemistry of Heterocyclic Compounds, 2023, 59 : 304 - 308
  • [4] The nitration and bromination of 2-(pentafluorosulfanyl)-1,3-benzothiazole and 2-(trifluoromethyl)-1,3-benzothiazole
    Guzyr, Olexandr I.
    Potikha, Lyudmila M.
    Shishkina, Svitlana V.
    Fetyukhin, Volodymyr N.
    Shermolovich, Yuriy G.
    CHEMISTRY OF HETEROCYCLIC COMPOUNDS, 2023, 59 (4-5) : 304 - 308
  • [5] Novel synthesis of pyrido[2,1-b]benzothiazoles and 1,3-benzothiazole derivatives
    Elgemeie, GH
    Shams, HZ
    Elkholy, YM
    Abbas, NS
    PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 2000, 165 : 265 - 272
  • [6] SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF 2-SUBSTITUTED BENZOTHIAZOLE DITHIOMIDOCARBONATE DERIVATIVES
    Tasleem
    INTERNATIONAL JOURNAL OF PHARMACEUTICAL SCIENCES AND RESEARCH, 2015, 6 (09): : 4058 - 4068
  • [7] NITRILES IN HETEROCYCLIC SYNTHESIS - NOVEL SYNTHESIS OF PYRIDO[2,1-B]BENZOTHIAZOLES AND 1,3-BENZOTHIAZOLE DERIVATIVES
    FATHY, NM
    MOTTI, FMA
    ELGEMEIE, GEH
    ARCHIV DER PHARMAZIE, 1988, 321 (09) : 509 - 512
  • [8] Synthesis, Characterization and Antifungal Activities of Amide and Acylthiourea of Substituted 2-Amino-1,3-Benzothiazole
    Wang, Junping
    Wang, Chuanping
    Wang, Hongmei
    Wei, Yan
    Lin, Jin
    Hao, Shuanghong
    NATURAL PRODUCT COMMUNICATIONS, 2025, 20 (01)
  • [9] 2,2′-(Sulfanediyldimethylene)bis(1,3-benzothiazole)
    Strasser, Christoph E.
    de Jongh, Leigh-Anne
    Raubenheimer, Helgard G.
    Cronje, Stephanie
    ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2011, 67 : O622 - U1745
  • [10] Synthesis and Antimicrobial Activity of Some New 2-Substituted Benzothiazole Derivatives
    Rajeeva, B.
    Srinivasulu, N.
    Shantakumar, S. M.
    E-JOURNAL OF CHEMISTRY, 2009, 6 (03) : 775 - 779
12345