Synthesis of 2,4-diaryl-2,3-dihydro-1,5-benzothiazepines as antibacterial and antifungal agents

被引：0
作者：
Barot, VM [1 ]
Patel, MR [1 ]
Naik, HB [1 ]
机构：
[1] Smt SMP Sci Coll, Dept Chem, Talod 383215, India
来源：
ASIAN JOURNAL OF CHEMISTRY | 2001年 / 13卷 / 01期
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
o-Aminophenol;reacts with chalcones (I) in methanol and acetic acid to give 3-(2-aminophenylmercapto)-3-amyl-propiophenones (II) which immediately undergo cyclisation in situ to give 2,4-diaryl-2,3-dihydro-1,5-benzothiazepines (IIIa).
引用
收藏
页码：347 / 349
页数：3
相关论文
共 50 条
[11]   SYNTHESIS OF 2, 4-DIARYL-2, 3-DIHYDRO-1, 5-BENZOTHIAZEPINES [J].
Ankodia, Vandana ;
Sharma, Praveen Kumar ;
Gupta, Vandana ;
Kumar, M. .
HETEROCYCLIC COMMUNICATIONS, 2008, 14 (03) :155-160
[12]   SYNTHESIS OF 2, 4-DIARYL-2, 3-DIHYDRO-1,5-BENZOTHIAZEPINES AND THEIR 1,1-DIOXIDES AS ANTI-BACTERIAL AGENTS [J].
JADHAV, KP ;
INGLE, DB .
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 1983, 22 (02) :180-182
[13]   An efficient procedure for the preparation of 3-acetyl-2,3-dihydrobenzothiazoles by ring contraction of 2,4-diaryl-2,3-dihydro-1,5-benzothiazepines under acetylating conditions [J].
Toth, G ;
Levai, A ;
Balazs, B ;
Simon, A .
LIEBIGS ANNALEN-RECUEIL, 1997, (05) :995-998
[14]   SYNTHESES OF 1,5-BENZOTHIAZEPINES .2. SYNTHESIS OF 4-ARYL-2-CARBOXY-2,3-DIHYDRO-1,5-BENZOTHIAZEPINES [J].
PANT, UC ;
GAUR, BS ;
CHUGH, M .
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 1987, 26 (10) :947-950
[15]   In silico studies on 2,3-dihydro-1,5-benzothiazepines as cholinesterase inhibitors [J].
Farzana Latif Ansari ;
Saima Kalsoom ;
Zahra Zaheer-ul-Haq ;
Farukh Ali .
Medicinal Chemistry Research, 2012, 21 :2329-2339
[16]   PREPARATION OF SUBSTITUTED 1H-2,3-DIHYDRO-1,5-BENZODIAZEPINES AND 2,3-DIHYDRO-1,5-BENZOTHIAZEPINES [J].
VOIGT, H .
ZEITSCHRIFT FUR CHEMIE, 1981, 21 (03) :102-103
[17]   In silico studies on 2,3-dihydro-1,5-benzothiazepines as cholinesterase inhibitors [J].
Ansari, Farzana Latif ;
Kalsoom, Saima ;
ul-Haq, Zaheer ;
Ali, Zahra ;
Jabeen, Farukh .
MEDICINAL CHEMISTRY RESEARCH, 2012, 21 (09) :2329-2339
[18]   Synthesis of 4-amino-3-dialkylaminomethyl-2,3-dihydro-1,5-benzothiazepines [J].
Yaccoubi, F ;
El Efrit, ML ;
Zantour, H .
PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 2002, 177 (10) :2321-2330
[19]   NEW HETEROCYCLIC SYSTEM SYNTHESIS H THE REACTION OF 2,3-DIHYDRO-1,5-BENZOTHIAZEPINES WITH DICHLOROCARBENE [J].
Ruo Xi LAN Sheng JIN Department of Chemistry .
ChineseChemicalLetters, 1992, (01) :9-10
[20]   Magnesium perchlorate as a new and highly efficient catalyst for the synthesis of 2,3-dihydro-1,5-benzothiazepines [J].
Khatik, Gopal L. ;
Kumar, Raj ;
Chakraborti, Asit K. .
SYNTHESIS-STUTTGART, 2007, (04) :541-546
12345