Synthesis and Insecticidal Evaluation of Novel N-Pyridylpyrazolecarboxamides Containing Different Substituents in the ortho-Position

被引：8

作者：

Feng Qi ^{[1
]}

Yu Guanping ^{[1
]}

Xiong Lixia ^{[1
]}

Wang Mingzhong ^{[1
]}

Li Zhengming ^{[1
]}

机构：

[1] Nankai Univ, State Key Lab Elementoorgan Chem, Inst Elementoorgan Chem, Tianjin 300071, Peoples R China

来源：

CHINESE JOURNAL OF CHEMISTRY | 2011年 / 29卷 / 08期

基金：

中国国家自然科学基金;

关键词：

insecticidal activity; N-pyridylpyrazole; pyrazolecarboxamide; ortho-substituents;

D O I：

10.1002/cjoc.201180295

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

In order to look for novel insecticides containing N-pyridylpyrazole, ten novel pyrazolecarboxamides containing different ortho-substituents in the aniline part were synthesized, and their structures were characterized by (1)H NMR, (13)C NMR and HRMS. The single crystal structure of 10b was determined by X-ray diffraction. Their evaluated insecticidal activity against oriental armyworm (Mythimna separata) indicated that all the compounds exhibited moderate insecticidal activities.

引用

页码：1651 / 1655

页数：5

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